Cloned (Comment) | Organism |
---|---|
expressed in COS-7 and Neuro2A cells | Mus musculus |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1-(tert-butyl)-3-(1-naphthyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | inhibits ATP analog-specific PKCdelta isoform | Mus musculus | |
1-(tert-butyl)-3-(2-methylbenzyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | inhibits ATP analog-specific PKCdelta isoform | Mus musculus | |
bisindolylmaleimide I | - |
Mus musculus | |
additional information | not inhibited by 1-tert-butyl-3-(2-naphthalenylmethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | Mus musculus | |
staurosporine | - |
Mus musculus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + a protein | Mus musculus | - |
ADP + phosphorylated protein | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Mus musculus | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + a protein | - |
Mus musculus | ADP + phosphorylated protein | - |
? | |
Nepsilon-(benzyl)-ATP + histone 3 | - |
Mus musculus | ADP + phosphorylated histone 3 | - |
? | |
Nepsilon-(benzyl)-ATP + RFARKGSLRQKNV | - |
Mus musculus | Nepsilon-(benzyl)-ADP + RFARKGpSLRQKNV | - |
? |
Synonyms | Comment | Organism |
---|---|---|
AS PKCdelta | - |
Mus musculus |
ATP analog specific protein kinase Cdelta | - |
Mus musculus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.000154 | - |
ATP analog-specific PKCdelta isoform, at pH 7.4 and 27°C | Mus musculus | 1-(tert-butyl)-3-(1-naphthyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine | |
0.000221 | - |
ATP analog-specific PKCdelta isoform, at pH 7.4 and 27°C | Mus musculus | bisindolylmaleimide I | |
0.00167 | - |
ATP analog-specific PKCdelta isoform, at pH 7.4 and 27°C | Mus musculus | staurosporine | |
0.0026 | - |
ATP analog-specific PKCdelta isoform, at pH 7.4 and 27°C | Mus musculus | 1-(tert-butyl)-3-(2-methylbenzyl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine |