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BRENDA support

Literature summary for 2.7.11.13 extracted from

  • Hegedus, C.; Lakatos, P.; Olah, G.; Toth, B.I.; Gergely, S.; Szabo, E.; Biro, T.; Szabo, C.; Virag, L.
    Protein kinase C protects from DNA damage-induced necrotic cell death by inhibiting poly(ADP-ribose) polymerase-1 (2008), FEBS Lett., 582, 1672-1678.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
phorbol 12-myristate 13-acetate 100 nM Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
GF109203X bisindolylmaleimide, broad spectrum PKC inhibitor Mus musculus
Go6976 inhibitor of conventional (calcium-dependent) PKC isoforms Mus musculus

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
thymocyte
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + poly(ADP-ribose) polymerase-1
-
Mus musculus ADP + phosphorylated poly(ADP-ribose) polymerase-1
-
?

Synonyms

Synonyms Comment Organism
PKC
-
Mus musculus
protein kinase C
-
Mus musculus