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Literature summary for 2.7.11.1 extracted from
- Precise design of highly isoform-selective p21-activated kinase 4 inhibitors computational insights into the selectivity mechanism through molecular dynamics simulation and binding free energy calculation (2020), J. Biomol. Struct. Dyn., 38, 3825-3837 .
Inhibitors
| Inhibitors | Comment | Organism | Structure |
|---|---|---|---|
| PF-3758309 | - |
Homo sapiens |
Organism
| Organism | UniProt | Comment | Textmining |
|---|---|---|---|
| Homo sapiens | O96013 | - |
- |
| Homo sapiens | Q13153 | - |
- |
Synonyms
| Synonyms | Comment | Organism |
|---|---|---|
| p21-activated kinase 4 | - |
Homo sapiens |
| Pak1 | - |
Homo sapiens |
| PAK4 | - |
Homo sapiens |
Ki Value [mM]
| Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
|---|---|---|---|---|---|
| 0.000015 | - |
PF-3758309 | pH and temperature not specified in the publication | Homo sapiens | |
| 0.000039 | - |
PF-3758309 | pH and temperature not specified in the publication | Homo sapiens |
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