Cloned (Comment) | Organism |
---|---|
expressed in Spodoptera frugiperda (Sf9) cells | Monosiga brevicollis |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
BIRB-796 | about 60% residual activity at 0.02 mM | Monosiga brevicollis | |
dasatinib | about 3% residual activity at 0.02 mM | Monosiga brevicollis | |
DSA-1 | about 10% residual activity at 0.02 mM | Monosiga brevicollis | |
DSA-8 | about 20% residual activity at 0.02 mM | Monosiga brevicollis | |
imatinib | about 80% residual activity at 0.02 mM | Monosiga brevicollis | |
MC25a | about 65% residual activity at 0.02 mM | Monosiga brevicollis | |
nilotinib | about 70% residual activity at 0.02 mM | Monosiga brevicollis | |
sorafenib | about 30% residual activity at 0.02 mM | Monosiga brevicollis | |
VX-680 | about 5% residual activity at 0.02 mM | Monosiga brevicollis |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.29 | - |
ATP | at pH 7.5 and 30°C | Monosiga brevicollis |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Monosiga brevicollis | - |
- |
- |
Purification (Comment) | Organism |
---|---|
Ni-NTA column chromatography | Monosiga brevicollis |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + EAIYAAPFAKKKG | - |
Monosiga brevicollis | ADP + EAI-pY-AAPFAKKKG | - |
? |
Synonyms | Comment | Organism |
---|---|---|
ABL2 | - |
Monosiga brevicollis |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.37 | - |
ATP | at pH 7.5 and 30°C | Monosiga brevicollis |