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Literature summary for 2.7.10.2 extracted from

  • Jongstra-Bilen, J.; Puig Cano, A.; Hasija, M.; Xiao, H.; Smith, C.I.; Cybulsky, M.I.
    Dual functions of Brutons tyrosine kinase and Tec kinase during Fcgamma receptor-induced signaling and phagocytosis (2008), J. Immunol., 181, 288-298.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information Btk activation is induced by FcgammaR signaling, activation requires binding to phosphatidylinositol 3,4,5-trisphosphate Mus musculus
additional information Tec activation is induced by FcgammaR signaling, activation requires binding to phosphatidylinositol 3,4,5-trisphosphate Mus musculus

Inhibitors

Inhibitors Comment Organism Structure
LFM-A13
-
Mus musculus
siRNA
-
Mus musculus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + [protein]-L-tyrosine Mus musculus
-
ADP + [protein]-L-tyrosine phosphate
-
?

Organism

Organism UniProt Comment Textmining
Mus musculus
-
-
-
Mus musculus P24604
-
-

Posttranslational Modification

Posttranslational Modification Comment Organism
phosphoprotein phosphorylation by other kinases and autophosphorylation Mus musculus
phosphoprotein phosphorylation by other kinases and autophosphorylation at Tyr223 of Btk Mus musculus

Source Tissue

Source Tissue Comment Organism Textmining
peritoneal macrophage
-
Mus musculus
-
RAW-264.7 cell
-
Mus musculus
-
splenocyte
-
Mus musculus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + [protein]-L-tyrosine
-
Mus musculus ADP + [protein]-L-tyrosine phosphate
-
?

Synonyms

Synonyms Comment Organism
Brutons tyrosine kinase
-
Mus musculus
Btk
-
Mus musculus
Tec kinase
-
Mus musculus