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Literature summary for 2.7.10.2 extracted from

  • Gao, Z.; Lau, C.P.; Wong, T.M.; Li, G.R.
    Protein tyrosine kinase-dependent modulation of voltage-dependent potassium channels by genistein in rat cardiac ventricular myocytes (2004), Cell. Signal., 16, 333-341.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
4-amino-5-(4-chlorophenyl)-7-(tert-butyl)pyrazolo[3,4-d] pyrimidine i.e. pp2, inhibits Src family PTKs Rattus norvegicus
genistein isoflavone, inhibits PTKs, and reversibly inhibits voltage-dependent transient outward and rectifier inward K+-currents in myocytes, overview Rattus norvegicus
tyrphostin A23 inhibits PTKs Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
cytosol Src family PTKs Rattus norvegicus 5829
-

Metals/Ions

Metals/Ions Comment Organism Structure
Mg2+
-
Rattus norvegicus

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
additional information Rattus norvegicus protein tyrosine kinase-dependent modulation of voltage-dependent potassium channels by genistein in cardiac ventricular myocytes ?
-
?

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
male sprague-dawley rats
-

Source Tissue

Source Tissue Comment Organism Textmining
heart
-
Rattus norvegicus
-
heart ventricle
-
Rattus norvegicus
-
myocyte ventricular Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
additional information protein tyrosine kinase-dependent modulation of voltage-dependent potassium channels by genistein in cardiac ventricular myocytes Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
Protein tyrosine kinase
-
Rattus norvegicus
PTK
-
Rattus norvegicus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
additional information
-
additional information
-
Rattus norvegicus