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Literature summary for 2.7.10.2 extracted from

  • Burlando, B.; Magnelli, V.; Panfoli, I.; Berti, E.; Viarengo, A.
    Ligand-independent tyrosine kinase signalling in RTH 149 trout hepatoma cells: comparison among heavy metals and pro-oxidants (2003), Cell. Physiol. Biochem., 13, 147-154.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
H2O2 increases tyrosine phosphorylation in vivo, genistein decreases the activating effect Oncorhynchus mykiss

Inhibitors

Inhibitors Comment Organism Structure
genistein
-
Oncorhynchus mykiss

Metals/Ions

Metals/Ions Comment Organism Structure
Cu2+ increases tyrosine phosphorylation in vivo, prevented by preincubation with genistein Oncorhynchus mykiss
Hg2+ increases tyrosine phosphorylation in vivo, genistein decreases the activating effect Oncorhynchus mykiss

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
ATP + a [protein]-L-tyrosine Oncorhynchus mykiss
-
ADP + a [protein]-L-tyrosine phosphate
-
?
additional information Oncorhynchus mykiss enzyme is involved in cell growth, differentiation, and apoptosis ?
-
?

Organism

Organism UniProt Comment Textmining
Oncorhynchus mykiss
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
hepatoma cell
-
Oncorhynchus mykiss
-
RTH-149 cell hepatoma cell line Oncorhynchus mykiss
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ATP + a [protein]-L-tyrosine
-
Oncorhynchus mykiss ADP + a [protein]-L-tyrosine phosphate
-
?
additional information enzyme is involved in cell growth, differentiation, and apoptosis Oncorhynchus mykiss ?
-
?

Synonyms

Synonyms Comment Organism
non-receptor tyrosine kinase
-
Oncorhynchus mykiss