Inhibitors | Comment | Organism | Structure |
---|---|---|---|
ADP | kinetics | Homo sapiens | |
CMP | - |
Homo sapiens | |
CTP | - |
Homo sapiens | |
Cytosine arabinoside monophosphate | strong | Homo sapiens | |
Cytosine arabinoside triphosphate | - |
Homo sapiens | |
dAMP | strong | Homo sapiens | |
dATP | strong | Homo sapiens | |
dCDP | - |
Homo sapiens | |
dCMP | product inhibition, strong | Homo sapiens | |
dCTP | kinetics | Homo sapiens | |
dGMP | strong | Homo sapiens | |
Dideoxyadenosine | - |
Homo sapiens | |
Dideoxycytidine | - |
Homo sapiens | |
dUMP | strong | Homo sapiens | |
dUTP | - |
Homo sapiens | |
GDP | - |
Homo sapiens | |
IMP | - |
Homo sapiens | |
P1,P4-diadenosine 5'-tetraphosphate | not di-, tri- or pentaphosphate derivative | Homo sapiens | |
Sodium diphosphate | not monophosphate | Homo sapiens | |
UDP | strong | Homo sapiens | |
UMP | strong | Homo sapiens | |
UTP | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | - |
Homo sapiens | |
0.0008 | 0.0015 | deoxycytidine | 37°C, pH 7.0 | Homo sapiens | |
0.02 | 0.04 | cytosine arabinoside | pH 7.0, 37°C | Homo sapiens | |
0.33 | 0.43 | deoxyguanosine | 37°C, pH 7.0 | Homo sapiens | |
0.45 | - |
cytidine | 37°C, pH 7.0 | Homo sapiens | |
0.5 | - |
deoxyadenosine | 37°C, pH 7.0 | Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | Mg2+/ATP complex is the reactive species | Homo sapiens | |
Mg2+ | maximal activity at a ATP:Mg2+-ratio of 1:1 | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
leukemia cell | leukemic T-lymphoblasts | Homo sapiens | - |
leukemia cell | cell line MOLT-4 | Homo sapiens | - |
MOLT-4 cell | - |
Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
8 | - |
37°C, pH 7.0 | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + 2'-deoxycytidine | - |
Homo sapiens | ADP + 5'-dCMP | - |
? | |
ATP + cytidine | - |
Homo sapiens | ADP + ? | - |
? | |
NTP + cytosine arabinoside | - |
Homo sapiens | NDP + cytosine arabinoside 5'-monophosphate | - |
? | |
NTP + deoxyadenosine | - |
Homo sapiens | NDP + dAMP | - |
? | |
NTP + deoxycytidine | enzyme shows little specificity towards phosphate donor | Homo sapiens | NDP + dCMP | - |
? | |
NTP + deoxyguanosine | - |
Homo sapiens | NDP + dGMP | - |
? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |