Activating Compound | Comment | Organism | Structure |
---|---|---|---|
Triton X-100 | - |
Saccharomyces cerevisiae |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
adenosine | inhibits in the millimolar range | Saccharomyces cerevisiae | |
Ca2+ | - |
Saccharomyces cerevisiae | |
Ly-294002 | IC50: 0.05-0.1 mM; IC50: 0.1 mM | Saccharomyces cerevisiae | |
additional information | insensitive to wortmannin and LY-294002 | Saccharomyces cerevisiae | |
Phenylarsine oxide | IC50: 0.001-0.005 mM; IC50: 0.03 mM; IC50: above 0.1 mM | Saccharomyces cerevisiae | |
Wortmannin | IC50: 0.05-0.3 mM; IC50: 50-300 nM | Saccharomyces cerevisiae |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.01 | 0.05 | ATP | - |
Saccharomyces cerevisiae | |
0.02 | 0.06 | 1-phosphatidyl-1D-myo-inositol | - |
Saccharomyces cerevisiae | |
0.1 | - |
1-phosphatidyl-1D-myo-inositol | - |
Saccharomyces cerevisiae | |
0.4 | - |
ATP | - |
Saccharomyces cerevisiae | |
0.7 | - |
ATP | - |
Saccharomyces cerevisiae |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
Golgi apparatus | - |
Saccharomyces cerevisiae | 5794 | - |
plasma membrane | - |
Saccharomyces cerevisiae | 5886 | - |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
additional information | no direct effect by Ca2+ | Saccharomyces cerevisiae |
Molecular Weight [Da] | Molecular Weight Maximum [Da] | Comment | Organism |
---|---|---|---|
54000 | - |
calculated from amino acid sequence | Saccharomyces cerevisiae |
55000 | - |
calculated from amino acid sequence | Saccharomyces cerevisiae |
92000 | - |
calculated from amino acid sequence | Saccharomyces cerevisiae |
230000 | - |
calculated from amino acid sequence | Saccharomyces cerevisiae |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Saccharomyces cerevisiae | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + 1-phosphatidyl-1D-myo-inositol | - |
Saccharomyces cerevisiae | ADP + 1-phosphatidyl-1D-myo-inositol 4-phosphate | - |
r |
Synonyms | Comment | Organism |
---|---|---|
56 kDa type II PtdIns 4-kinase | - |
Saccharomyces cerevisiae |
Lsb6p | - |
Saccharomyces cerevisiae |
phosphatidylinositol 4-kinase | - |
Saccharomyces cerevisiae |
Pik1p | - |
Saccharomyces cerevisiae |
PIK230 | - |
Saccharomyces cerevisiae |
Pik2p | - |
Saccharomyces cerevisiae |
Pik4ca | - |
Saccharomyces cerevisiae |
PIK4IIalpha | - |
Saccharomyces cerevisiae |
PIK4IIbeta | - |
Saccharomyces cerevisiae |
PIK4IIIalpha | - |
Saccharomyces cerevisiae |
PIK4IIIbeta | - |
Saccharomyces cerevisiae |
PIK55 | - |
Saccharomyces cerevisiae |
PtdIns 4-kinase | - |
Saccharomyces cerevisiae |
PtdIns 4-kinase beta | - |
Saccharomyces cerevisiae |
Stt4p | - |
Saccharomyces cerevisiae |
Cofactor | Comment | Organism | Structure |
---|---|---|---|
ATP | - |
Saccharomyces cerevisiae |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.01 | 0.07 | adenosine | - |
Saccharomyces cerevisiae |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00005 | 0.0003 | IC50: 50-300 nM | Saccharomyces cerevisiae | Wortmannin | |
0.001 | 0.005 | IC50: 0.001-0.005 mM | Saccharomyces cerevisiae | Phenylarsine oxide | |
0.03 | - |
IC50: 0.03 mM | Saccharomyces cerevisiae | Phenylarsine oxide | |
0.05 | 0.1 | IC50: 0.05-0.1 mM | Saccharomyces cerevisiae | Ly-294002 | |
0.05 | 0.3 | IC50: 0.05-0.3 mM | Saccharomyces cerevisiae | Wortmannin | |
0.1 | - |
IC50: 0.1 mM | Saccharomyces cerevisiae | Ly-294002 | |
0.1 | - |
IC50: above 0.1 mM | Saccharomyces cerevisiae | Phenylarsine oxide |