Any feedback?
Please rate this page
(literature.php)
(0/150)

BRENDA support

Literature summary for 2.7.1.40 extracted from

  • Lepper, T.W.; Oliveira, E.; Koch, G.D.; Berlese, D.B.; Feksa, L.R.
    Lead inhibits in vitro creatine kinase and pyruvate kinase activity in brain cortex of rats (2009), Toxicol. In Vitro, 24, 1045-1051.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
additional information cysteamine or glutathione per se do not modify enzymatic activity, but prevent the toxic effects of lead Rattus norvegicus
Pb2+ lead inhibits pyruvate kinase activity in a dose-dependent manner by interaction with its thiol groups Rattus norvegicus

Localization

Localization Comment Organism GeneOntology No. Textmining
cytosol
-
Rattus norvegicus 5829
-

Organism

Organism UniProt Comment Textmining
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain cortex cell line
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
ADP + phosphoenolpyruvate
-
Rattus norvegicus ATP + pyruvate
-
?

Synonyms

Synonyms Comment Organism
ATP:pyruvate 2-O-phosphotransferase
-
Rattus norvegicus

Cofactor

Cofactor Comment Organism Structure
ADP
-
Rattus norvegicus