Inhibitors | Comment | Organism | Structure |
---|---|---|---|
NSC 122612 | 0.12 mM, 27% inhibition | Escherichia coli | |
NSC 19791 | 0.89 mM, 14% inhibition | Escherichia coli | |
NSC 23145 | 0.105 mM, 23% inhibition | Escherichia coli | |
NSC 298251 | 0.1 mM, 30% inhibition | Escherichia coli | |
NSC 3056 | 0.089 mM, 24% inhibition | Escherichia coli | |
NSC 309091 | 0.13 mM, 21% inhibition | Escherichia coli | |
NSC 357688 | 0.09 mM, 28% inhibition | Escherichia coli | |
NSC 43275 | 0.106 mM, 16% inhibition | Escherichia coli | |
NSC 6487 | 0.089 mM, 6% inhibition | Escherichia coli | |
NSC 65043 | 0.093 mM, 84% inhibition, linear competitive | Escherichia coli | |
NSC 65043 | IC50: 0.077 mM | Homo sapiens | |
NSC 659977 | 0.134 mM, 60% inhibition | Escherichia coli | |
NSC 81031 | 0.93 mM, 15% inhibition | Escherichia coli |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Escherichia coli | - |
- |
- |
Homo sapiens | - |
recombinant enzyme | - |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
2 | 5 | NSC 65043 | - |
Homo sapiens | |
12.5 | - |
NSC 65043 | - |
Escherichia coli |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.077 | - |
IC50: 0.077 mM | Homo sapiens | NSC 65043 |