Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(2-tert-butoxy-2-oxoethyl)(dimethyl)sulfonium | - |
Homo sapiens | |
(2-[[(1R)-3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-1-carboxy-3-oxopropyl]amino]-2-oxoethyl)(dimethyl)sulfanium bromide | - |
Homo sapiens | |
(2-[[4-(methoxycarbonyl)benzyl]oxy]-2-oxoethyl)(dimethyl)sulfonium | - |
Homo sapiens | |
(2-[[6-(methoxycarbonyl)naphthalen-2-yl]methoxy]-2-oxoethyl)(dimethyl)sulfonium | - |
Homo sapiens | |
(naphthalen-2-yl)methyl 4-(N-acryloylglycyl)piperazine-1-carboxylate | - |
Homo sapiens | |
(naphthalen-2-yl)methyl 4-[N-(bromoacetyl)glycyl]piperazine-1-carboxylate | - |
Homo sapiens | |
1-(ethenylsulfonyl)tricyclo[3.3.1.13,7]decane | - |
Homo sapiens | |
1-(tricyclo[3.3.1.13,7]dec-1-yl)prop-2-en-1-one | - |
Homo sapiens | |
2-(tricyclo[3.3.1.13,7]dec-1-yl)ethyl prop-2-enoate | - |
Homo sapiens | |
2-([2-[(3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-2,3-dioxopropyl)amino]-2-oxoethyl]sulfanyl)-1,3,4,5-tetramethyl-1H-imidazol-3-ium bromide | - |
Homo sapiens | |
2-bromo-1-(tricyclo[3.3.1.13,7]dec-1-yl)ethanone | - |
Homo sapiens | |
2-chloro-1-(tricyclo[3.3.1.13,7]dec-1-yl)ethanone | - |
Homo sapiens | |
benzyl 4-[3-(acryloylamino)-2-oxopropanoyl]piperazine-1-carboxylate | - |
Homo sapiens | |
benzyl 4-[3-[(ethenylsulfonyl)amino]-2-oxopropanoyl]piperazine-1-carboxylate | - |
Homo sapiens | |
dimethyl[2-oxo-2-(tricyclo[3.3.1.13,7]dec-1-yl)ethyl]sulfonium | - |
Homo sapiens | |
dimethyl[2-oxo-2-(tricyclo[3.3.1.13,7]dec-1-ylmethoxy)ethyl]sulfonium | - |
Homo sapiens | |
dimethyl[2-oxo-2-[2-(tricyclo[3.3.1.13,7]dec-1-yl)ethoxy]ethyl]sulfonium | - |
Homo sapiens | |
methyl 4-[(acryloyloxy)methyl]benzoate | - |
Homo sapiens | |
methyl 4-[[(bromoacetyl)oxy]methyl]benzoate | - |
Homo sapiens | |
methyl 6-[(acryloyloxy)methyl]naphthalene-2-carboxylate | - |
Homo sapiens | |
methyl 6-[[(bromoacetyl)oxy]methyl]naphthalene-2-carboxylate | - |
Homo sapiens | |
methyl 6-[[(chloroacetyl)oxy]methyl]naphthalene-2-carboxylate | - |
Homo sapiens | |
N-(2-[4-[5-(dimethylamino)naphthalene-1-sulfonyl]piperazin-1-yl]-2-oxoethyl)prop-2-enamide | - |
Homo sapiens | |
tricyclo[3.3.1.13,7]dec-1-ylmethyl bromoacetate | - |
Homo sapiens | |
tricyclo[3.3.1.13,7]dec-1-ylmethyl prop-2-enoate | - |
Homo sapiens | |
[2-[(2-[4-[5-(dimethylamino)naphthalene-1-sulfonyl]piperazin-1-yl]-2-oxoethyl)amino]-2-oxoethyl](dimethyl)sulfanium | - |
Homo sapiens | |
[2-[(3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-2,3-dioxopropyl)amino]-2-oxoethyl](diethyl)sulfanium bromide | - |
Homo sapiens | |
[2-[(3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-2,3-dioxopropyl)amino]-2-oxoethyl](dimethyl)sulfanium bromide | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
HUVEC cell | - |
Homo sapiens | - |
NIH-3T3 cell | - |
Homo sapiens | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
Cbz-Gln-Gly + alkylamine | - |
Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
TG2 | - |
Homo sapiens |
transglutaminase | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0000021 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | methyl 4-[[(bromoacetyl)oxy]methyl]benzoate | |
0.0000039 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | 2-bromo-1-(tricyclo[3.3.1.13,7]dec-1-yl)ethanone | |
0.0000061 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | N-(2-[4-[5-(dimethylamino)naphthalene-1-sulfonyl]piperazin-1-yl]-2-oxoethyl)prop-2-enamide | |
0.00000629 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | tricyclo[3.3.1.13,7]dec-1-ylmethyl bromoacetate | |
0.00000665 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | methyl 6-[[(chloroacetyl)oxy]methyl]naphthalene-2-carboxylate | |
0.00000875 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | 2-chloro-1-(tricyclo[3.3.1.13,7]dec-1-yl)ethanone | |
0.000015 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | methyl 6-[[(bromoacetyl)oxy]methyl]naphthalene-2-carboxylate | |
0.000029 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (naphthalen-2-yl)methyl 4-[N-(bromoacetyl)glycyl]piperazine-1-carboxylate | |
0.000125 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | 1-(tricyclo[3.3.1.13,7]dec-1-yl)prop-2-en-1-one | |
0.000273 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (2-tert-butoxy-2-oxoethyl)(dimethyl)sulfonium | |
0.00038 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | [2-[(2-[4-[5-(dimethylamino)naphthalene-1-sulfonyl]piperazin-1-yl]-2-oxoethyl)amino]-2-oxoethyl](dimethyl)sulfanium | |
0.00044 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (naphthalen-2-yl)methyl 4-(N-acryloylglycyl)piperazine-1-carboxylate | |
0.0007 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (2-[[(1R)-3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-1-carboxy-3-oxopropyl]amino]-2-oxoethyl)(dimethyl)sulfanium bromide | |
0.000775 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | dimethyl[2-oxo-2-(tricyclo[3.3.1.13,7]dec-1-ylmethoxy)ethyl]sulfonium | |
0.000875 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | 1-(ethenylsulfonyl)tricyclo[3.3.1.13,7]decane | |
0.000889 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | dimethyl[2-oxo-2-(tricyclo[3.3.1.13,7]dec-1-yl)ethyl]sulfonium | |
0.0009 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | 2-(tricyclo[3.3.1.13,7]dec-1-yl)ethyl prop-2-enoate | |
0.00107 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (naphthalen-2-yl)methyl 4-(N-acryloylglycyl)piperazine-1-carboxylate | |
0.0014 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | [2-[(3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-2,3-dioxopropyl)amino]-2-oxoethyl](dimethyl)sulfanium bromide | |
0.0015 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (2-[[6-(methoxycarbonyl)naphthalen-2-yl]methoxy]-2-oxoethyl)(dimethyl)sulfonium | |
0.001625 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | tricyclo[3.3.1.13,7]dec-1-ylmethyl prop-2-enoate | |
0.001725 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | benzyl 4-[3-[(ethenylsulfonyl)amino]-2-oxopropanoyl]piperazine-1-carboxylate | |
0.00185 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | [2-[(3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-2,3-dioxopropyl)amino]-2-oxoethyl](diethyl)sulfanium bromide | |
0.0021 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | methyl 6-[(acryloyloxy)methyl]naphthalene-2-carboxylate | |
0.00315 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | dimethyl[2-oxo-2-[2-(tricyclo[3.3.1.13,7]dec-1-yl)ethoxy]ethyl]sulfonium | |
0.0033 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | (2-[[4-(methoxycarbonyl)benzyl]oxy]-2-oxoethyl)(dimethyl)sulfonium | |
0.005925 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | benzyl 4-[3-(acryloylamino)-2-oxopropanoyl]piperazine-1-carboxylate | |
0.0063 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | methyl 4-[(acryloyloxy)methyl]benzoate | |
0.1 | - |
at pH 7.1, temperature not specified in the publication | Homo sapiens | 2-([2-[(3-[4-[(benzyloxy)carbonyl]piperazin-1-yl]-2,3-dioxopropyl)amino]-2-oxoethyl]sulfanyl)-1,3,4,5-tetramethyl-1H-imidazol-3-ium bromide |