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Literature summary for 2.3.2.13 extracted from

  • Kawashima, S.
    Inhibition of rat liver transglutaminase by nucleotides (1991), Experientia, 47, 709-712.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
ADP complete inhibition of rat liver and human brain transglutaminase, reversible, non-competitive to putrescine Homo sapiens
ADP complete inhibition of rat liver and human brain transglutaminase, reversible, non-competitive to putrescine Rattus norvegicus
AMP weak inhibition of liver transglutaminase Rattus norvegicus
ATP 3 mM, complete inhibition of rat liver and human brain tissue-type transglutaminase, reversible; 3 mM, complete inhibition of rat liver and human brain transglutaminase, reversible, non-competitive to putrescine Homo sapiens
ATP 3 mM, complete inhibition of rat liver and human brain tissue-type transglutaminase, reversible; 3 mM, complete inhibition of rat liver and human brain transglutaminase, reversible, non-competitive to putrescine Rattus norvegicus
CTP 3 mM, complete inhibition of rat liver and human brain transglutaminase, reversible, non-competitive to putrescine Homo sapiens
CTP 3 mM, complete inhibition of rat liver and human brain transglutaminase, reversible, non-competitive to putrescine Rattus norvegicus
GTP 50% as effective as ATP Homo sapiens
GTP 50% as effective as ATP Rattus norvegicus
additional information
-
Homo sapiens
additional information not inhibited by adenosine or adenine Rattus norvegicus
UTP 50% as effective as ATP Rattus norvegicus

Metals/Ions

Metals/Ions Comment Organism Structure
Ca2+ requirement Homo sapiens
Ca2+ requirement Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Rattus norvegicus
-
tissue-type transglutaminase, abbrevation TGC
-

Purification (Commentary)

Purification (Comment) Organism
partial Homo sapiens
tissue-type transglutaminase Rattus norvegicus

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Homo sapiens
-
brain
-
Rattus norvegicus
-
liver
-
Homo sapiens
-
liver
-
Rattus norvegicus
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
putrescine + N,N'-dimethylcasein
-
Homo sapiens ?
-
?
putrescine + N,N'-dimethylcasein
-
Rattus norvegicus ?
-
?

Synonyms

Synonyms Comment Organism
transglutaminase C
-
Rattus norvegicus

Temperature Optimum [°C]

Temperature Optimum [°C] Temperature Optimum Maximum [°C] Comment Organism
37
-
assay at Homo sapiens
37
-
assay at Rattus norvegicus