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Literature summary for 2.3.1.48 extracted from

  • Mai, A.; Rotili, D.; Tarantino, D.; Nebbioso, A.; Castellano, S.; Sbardella, G.; Tini, M.; Altucci, L.
    Identification of 4-hydroxyquinolines inhibitors of p300/CBP histone acetyltransferases (2009), Bioorg. Med. Chem. Lett., 19, 1132-1135.
    View publication on PubMed
Search for more literature for 2.3.1.48

Inhibitors

Inhibitors Comment Organism Structure
(2R,3S)-4-methylidene-5-oxo-2-propyltetrahydrofuran-3-carboxylic acid i.e. butyrolactone MB-3, a GCN5 inhibitor Homo sapiens
2-decyl-4-hydroxyquinoline-3-carboxylic acid
-
 Homo sapiens
4-hydroxy-2-methylquinoline-3-carboxylic acid
-
 Homo sapiens
4-hydroxy-2-pentadecylquinoline-3-carboxylic acid
-
 Homo sapiens
4-hydroxy-2-pentylquinoline-3-carboxylic acid
-
 Homo sapiens
anacardic acid
-
 Homo sapiens
ethyl 2-decyl-4-hydroxyquinoline-3-carboxylate
-
 Homo sapiens
ethyl 4-hydroxy-2-methylquinoline-3-carboxylate
-
 Homo sapiens
ethyl 4-hydroxy-2-pentadecylquinoline-3-carboxylate
-
 Homo sapiens
ethyl 4-hydroxy-2-pentylquinoline-3-carboxylate
-
 Homo sapiens
additional information relative inhibition of p300, CBP, GCN5, and PCAF, overview Homo sapiens

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
U-937 cell
-
 Homo sapiens
-

Synonyms

Synonyms Comment Organism
Cbp
-
 Homo sapiens
Gcn5
-
 Homo sapiens
HAT
-
 Homo sapiens
p300/CBP histone acetyltransferase
-
 Homo sapiens
PCAF
-
 Homo sapiens