Activating Compound | Comment | Organism | Structure |
---|---|---|---|
1-hexadecyl-3-(trifluoroethyl)-sn-glycero-2-phosphomethanol | 20 microM, 149% of initial activity for detergent-solubilized enzyme | Caldalkalibacillus thermarum | |
17-beta-hydroxy-17-alpha-ethynyl-delta-4-androstano[3,2-b]pyrimido[1,2-a]benzimidazole | 20 microM, 142% of initial activity for detergent-solubilized enzyme | Caldalkalibacillus thermarum | |
2,6-difluoro-4-[2-(phenylsulfonylamino)ethylthio]phenoxyacetamide | 20 microM, 136% of initial activity for detergent-solubilized enzyme, 134% of initial activity for lipid-reconstituted enzyme | Caldalkalibacillus thermarum | |
pentylenetetrazole | 20 microM, 132% of initial activity for detergent-solubilized enzyme | Caldalkalibacillus thermarum |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
mangostin | 20 microM, 19% residual activity for detergent-solubilized enzyme | Caldalkalibacillus thermarum | |
morin | 20 microM, 32% residual activity for detergent-solubilized enzyme, 18.7% residual activity for lipid-reconstituted enzyme | Caldalkalibacillus thermarum | |
nordihydroguaiaretic acid | 20 microM, 33% residual activity for detergent-solubilized enzyme, 18.7% residual activity for lipid-reconstituted enzyme | Caldalkalibacillus thermarum | |
piceatannol | 20 microM, 35% residual activity for detergent-solubilized enzyme | Caldalkalibacillus thermarum | |
tyrphostin AG 537 | 20 microM, 22% residual activity for detergent-solubilized enzyme, 57% residual activity for lipid-reconstituted enzyme | Caldalkalibacillus thermarum | |
tyrphostin AG 808 | 20 microM, 7% residual activity for detergent-solubilized enzyme | Caldalkalibacillus thermarum |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Caldalkalibacillus thermarum | F5L3B8 | - |
- |
Caldalkalibacillus thermarum TA2.A1 | F5L3B8 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
NADH + H+ + menadione | - |
Caldalkalibacillus thermarum | NAD+ + menadiol | - |
? | |
NADH + H+ + menadione | - |
Caldalkalibacillus thermarum TA2.A1 | NAD+ + menadiol | - |
? |