Inhibitors | Comment | Organism | Structure |
---|---|---|---|
warfarin | IC50: 0.00007 mM | Bos taurus | |
warfarin | - |
Canis lupus familiaris | |
warfarin | - |
Equus caballus | |
warfarin | IC50: 0.00018 mM, only one sample measured | Homo sapiens | |
warfarin | IC50: 0.00017 mM | Mus musculus | |
warfarin | - |
Ovis aries | |
warfarin | IC50: 0.00012 mM, only one sample measured | Sus scrofa |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00241 | - |
vitamin K1 2,3-epoxide | 37°C | Ovis aries | |
0.00241 | - |
vitamin K1 2,3-epoxide | 37°C | Equus caballus | |
0.00309 | - |
vitamin K1 2,3-epoxide | 37°C, only one sample measured | Homo sapiens | |
0.0032 | - |
vitamin K1 2,3-epoxide | 37°C, only one sample measured | Sus scrofa | |
0.0036 | - |
vitamin K1 2,3-epoxide | 37°C | Canis lupus familiaris | |
0.00416 | - |
vitamin K1 2,3-epoxide | 37°C | Mus musculus | |
0.00425 | - |
vitamin K1 2,3-epoxide | 37°C | Bos taurus | |
0.00646 | - |
vitamin K1 2,3-epoxide | 37°C | Bos taurus |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
microsome | - |
Mus musculus | - |
- |
microsome | - |
Homo sapiens | - |
- |
microsome | - |
Sus scrofa | - |
- |
microsome | - |
Bos taurus | - |
- |
microsome | - |
Ovis aries | - |
- |
microsome | - |
Canis lupus familiaris | - |
- |
microsome | - |
Equus caballus | - |
- |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Bos taurus | - |
- |
- |
Canis lupus familiaris | - |
- |
- |
Equus caballus | - |
- |
- |
Homo sapiens | - |
- |
- |
Mus musculus | - |
- |
- |
Ovis aries | - |
- |
- |
Sus scrofa | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
liver | - |
Mus musculus | - |
liver | - |
Homo sapiens | - |
liver | - |
Sus scrofa | - |
liver | - |
Bos taurus | - |
liver | - |
Ovis aries | - |
liver | - |
Canis lupus familiaris | - |
liver | - |
Equus caballus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
vitamin K1 2,3-epoxide + dithiothreitol | - |
Mus musculus | vitamin K1 + oxidized dithiothreitol | - |
? | |
vitamin K1 2,3-epoxide + dithiothreitol | - |
Homo sapiens | vitamin K1 + oxidized dithiothreitol | - |
? | |
vitamin K1 2,3-epoxide + dithiothreitol | - |
Sus scrofa | vitamin K1 + oxidized dithiothreitol | - |
? | |
vitamin K1 2,3-epoxide + dithiothreitol | - |
Bos taurus | vitamin K1 + oxidized dithiothreitol | - |
? | |
vitamin K1 2,3-epoxide + dithiothreitol | - |
Ovis aries | vitamin K1 + oxidized dithiothreitol | - |
? | |
vitamin K1 2,3-epoxide + dithiothreitol | - |
Canis lupus familiaris | vitamin K1 + oxidized dithiothreitol | - |
? | |
vitamin K1 2,3-epoxide + dithiothreitol | - |
Equus caballus | vitamin K1 + oxidized dithiothreitol | - |
? |
Synonyms | Comment | Organism |
---|---|---|
VKOR | - |
Mus musculus |
VKOR | - |
Homo sapiens |
VKOR | - |
Sus scrofa |
VKOR | - |
Bos taurus |
VKOR | - |
Ovis aries |
VKOR | - |
Canis lupus familiaris |
VKOR | - |
Equus caballus |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Mus musculus |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Homo sapiens |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Sus scrofa |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Bos taurus |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Ovis aries |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Canis lupus familiaris |
warfarin-sensitive vitamin K1 2,3-epoxide reductase | - |
Equus caballus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00007 | - |
IC50: 0.00007 mM | Bos taurus | warfarin | |
0.00012 | - |
IC50: 0.00012 mM, only one sample measured | Sus scrofa | warfarin | |
0.00017 | - |
IC50: 0.00017 mM | Mus musculus | warfarin | |
0.00018 | - |
IC50: 0.00018 mM, only one sample measured | Homo sapiens | warfarin |