Inhibitors | Comment | Organism | Structure |
---|---|---|---|
1,10-Diaminodecane | 94% of initial activity at 2 mM | Rattus norvegicus | |
1,3-diaminopropane | 86% of initial activity at 0.5 mM | Rattus norvegicus | |
1,6-diaminohexane | 97% of initial activity at 2 mM | Rattus norvegicus | |
1,7-Diaminoheptane | 91% of initial activity at 2 mM | Rattus norvegicus | |
1,8-diaminooctane | 93% of initial activity at 2 mM | Rattus norvegicus | |
cadaverine | 87% of initial activity at 0.5 mM | Rattus norvegicus | |
caldine | 47% of initial activity at 0.5 mM | Rattus norvegicus | |
Lys-Thr-Gly-deoxyhypusine-His-Gly-His-Ala-Lys | competitive inhibition | Cricetulus griseus | |
additional information | no inhibition at 2 mM N-(2-cyanopropyl)-3-cyanopropylamine | Rattus norvegicus | |
N-(2-cyanoethyl)butane-1,4-diamine | 80% of initial activity at 2 mM | Rattus norvegicus | |
N-(3-cyanopropyl)propane-1,3-diamine | 79% of initial activity at 2 mM | Rattus norvegicus | |
putrescine | 85% of initial activity at 0.5 mM | Rattus norvegicus | |
spermidine | 58% of initial activity at 0.5 mM | Rattus norvegicus | |
spermine | 41% of initial activity at 0.5 mM | Rattus norvegicus | |
thermine | 35% of initial activity at 0.5 mM | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cricetulus griseus | - |
- |
- |
Rattus norvegicus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
ovary | - |
Cricetulus griseus | - |
testis | - |
Rattus norvegicus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
N'-(4-aminobutyl)lysine + electron donor + O2 | i.e. deoxyhypusine | Cricetulus griseus | N'-(4-amino-2-hydroxybutyl)lysine + oxidized electron donor + H2O | i.e. hypusine | ? | |
N'-(4-aminobutyl)lysine + electron donor + O2 | i.e. deoxyhypusine | Rattus norvegicus | N'-(4-amino-2-hydroxybutyl)lysine + oxidized electron donor + H2O | i.e. hypusine | ? |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Rattus norvegicus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7 | 7.5 | in 20 mM Tris buffer | Rattus norvegicus |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.25 | - |
spermine | competitive inhibition | Rattus norvegicus | |
0.44 | - |
Lys-Thr-Gly-deoxyhypusine-His-Gly-His-Ala-Lys | competitive inhibition | Cricetulus griseus |