Inhibitors | Comment | Organism | Structure |
---|---|---|---|
(R,S)-2-amino-oxo-4-(3'-4'-dichlorophenyl)butanoic acid | - |
Rattus norvegicus | |
3,4-dimethoxy-N-[4-(3-nitrophenyl)thiazol-2-yl]benzenesulfonamide | Ro-61-8048, 50% inhibition at 37 nM | Rattus norvegicus | |
4-amino-N-[4-[2-fluoro-5-(trifluoromethyl)phenyl]thiazol-2-yl]benzenesulfonamide | 50% inhibition at 19nM | Rattus norvegicus | |
additional information | inhibition by N-(4-phenylthiazol-2-yl)benzenesulfonamides with various modifications | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Rattus norvegicus | - |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000048 | - |
3,4-dimethoxy-N-[4-(3-nitrophenyl)thiazol-2-yl]benzenesulfonamide | competitive inhibitor | Rattus norvegicus | |
0.000095 | - |
(R,S)-2-amino-oxo-4-(3'-4'-dichlorophenyl)butanoic acid | competitive inhibitor | Rattus norvegicus |