Cloned (Comment) | Organism |
---|---|
recombinant human PHD2 (corresponding to residues 178-426 of the full-length PHD2 sequence) is expressed as a GST-fusion protein in Escherichia coli | Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.001 | - |
DLDLEALAPYIPADDDFQL | substrate: CODD peptide, pH 7, 37°C, without NaCl | Homo sapiens | |
0.001 | - |
DALTLLAPAAGDTIISLDYG | substrate: NODD peptide, pH 7, 37°C, without NaCl | Homo sapiens | |
0.0042 | - |
DLDLEALAPYIPADDDFQL | substrate: CODD peptide, pH 7, 37°C, 100 mM NaCl | Homo sapiens | |
0.0042 | - |
DALTLLAPAAGDTIISLDYG | substrate: NODD peptide, pH 7, 37°C, 100 mM NaCl | Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
NaCl | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
DALTLLAPAAGDTIISLDYG + 2-oxoglutarate + O2 | NODD peptide derived from native HIF-1alpha395-414 | Homo sapiens | ? | - |
? | |
DLDLEALAPYIPADDDFQL + 2-oxoglutarate + O2 | CODD peptide derived from native HIF-1alpha556-574. PHD2 preferred CODD by 20fold over NODD | Homo sapiens | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PHD2 | - |
Homo sapiens |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0101 | - |
DALTLLAPAAGDTIISLDYG | substrate: NODD peptide, pH 7, 37°C, without NaCl | Homo sapiens | |
0.0103 | - |
DALTLLAPAAGDTIISLDYG | substrate: NODD peptide, pH 7, 37°C, 100 mM NaCl | Homo sapiens | |
0.0188 | - |
DLDLEALAPYIPADDDFQL | substrate: CODD peptide, pH 7, 37°C, without NaCl | Homo sapiens | |
0.02 | - |
DLDLEALAPYIPADDDFQL | substrate: CODD peptide, pH 7, 37°C, 100 mM NaCl | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7 | - |
assay at | Homo sapiens |
kcat/KM Value [1/mMs-1] | kcat/KM Value Maximum [1/mMs-1] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
2.45 | - |
DALTLLAPAAGDTIISLDYG | substrate: NODD peptide, pH 7, 37°C, 100 mM NaCl | Homo sapiens | |
4.76 | - |
DLDLEALAPYIPADDDFQL | substrate: CODD peptide, pH 7, 37°C, 100 mM NaCl | Homo sapiens | |
10.1 | - |
DALTLLAPAAGDTIISLDYG | substrate: NODD peptide, pH 7, 37°C, without NaCl | Homo sapiens | |
18.8 | - |
DLDLEALAPYIPADDDFQL | substrate: CODD peptide, pH 7, 37°C, without NaCl | Homo sapiens |