Cloned (Comment) | Organism |
---|---|
expression in CHO cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
2-iodomelatonin | - |
Homo sapiens | |
2-iodomelatonin | - |
Mesocricetus auratus | |
5-methoxycarbonylamino-N-acetyltryptamine | - |
Homo sapiens | |
5-methoxycarbonylamino-N-acetyltryptamine | - |
Mesocricetus auratus | |
dicoumarol | - |
Homo sapiens | |
dicoumarol | - |
Mesocricetus auratus | |
Melatonin | - |
Homo sapiens | |
Melatonin | - |
Mesocricetus auratus | |
N-acetylserotonin | - |
Homo sapiens | |
N-acetylserotonin | - |
Mesocricetus auratus | |
S26553 | - |
Homo sapiens | |
S26553 | i.e. N-methyl-[1-[2-(acetylamino)ethyl]naphthalen-7-yl]-carbamate | Mesocricetus auratus | |
serotonin | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0089 | - |
menadione | pH 7.5 | Homo sapiens | |
0.0252 | - |
menadione | pH 7.5 | Mesocricetus auratus | |
0.0576 | - |
dihydrobenzylnicotinamide | pH 7.5 | Homo sapiens | |
0.0608 | - |
dihydrobenzylnicotinamide | pH 7.5 | Mesocricetus auratus |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
additional information | Homo sapiens | enzyme exhibits melatonin-binding activity | ? | - |
? | |
additional information | Mesocricetus auratus | enzyme exhibits melatonin-binding activity | ? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
expressed in CHO cells | - |
Mesocricetus auratus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
- |
Homo sapiens |
- |
Mesocricetus auratus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
kidney | - |
Homo sapiens | - |
kidney | - |
Mesocricetus auratus | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
menadione + dihydrobenzylnicotinamide | - |
Homo sapiens | ? | - |
? | |
menadione + dihydrobenzylnicotinamide | - |
Mesocricetus auratus | ? | - |
? | |
additional information | enzyme exhibits melatonin-binding activity | Homo sapiens | ? | - |
? | |
additional information | enzyme exhibits melatonin-binding activity | Mesocricetus auratus | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
melatonin-binding site MT3 | - |
Homo sapiens |
melatonin-binding site MT3 | - |
Mesocricetus auratus |
QR2 | - |
Homo sapiens |
quinone reductase 2 | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0012 | - |
2-iodomelatonin | pH 7.5 | Mesocricetus auratus | |
0.0028 | - |
S26553 | pH 7.5 | Mesocricetus auratus | |
0.029 | - |
2-iodomelatonin | pH 7.5 | Homo sapiens | |
0.0414 | - |
S26553 | pH 7.5 | Homo sapiens | |
0.043 | - |
Melatonin | pH 7.5 | Mesocricetus auratus | |
0.0435 | - |
5-methoxycarbonylamino-N-acetyltryptamine | pH 7.5 | Mesocricetus auratus | |
0.092 | - |
N-acetylserotonin | pH 7.5 | Mesocricetus auratus | |
0.204 | - |
N-acetylserotonin | pH 7.5 | Homo sapiens | |
0.246 | - |
Melatonin | pH 7.5 | Homo sapiens | |
0.376 | - |
5-methoxycarbonylamino-N-acetyltryptamine | pH 7.5 | Homo sapiens | |
0.566 | - |
dicoumarol | pH 7.5 | Mesocricetus auratus | |
0.62 | - |
dicoumarol | pH 7.5 | Homo sapiens | |
2.933 | - |
serotonin | - |
Homo sapiens |