0.5 mM significantly reduce the P-glycoprotein protein expression, 0.1 mM of 1-monoolein does not have any significant effect on the expression of P-glycoprotein
0.5 mM significantly reduce the P-glycoprotein protein expression, 0.1 mM of 1-monostearin does not have any significant effect on the expression of P-glycoprotein
flippase activity for 1-oleoyl-2-[6-(7-nitrol-2-1,3-benzonadiol-4-yl)amino]-sn-glycerophosphoethanolamine is inhibited by 72% at 5 mM 4-(2-aminoethyl)benzenesulfonyl fluoride, flippase activity for 1-oleoyl-2-[6-(7-nitrol-2-1,3-benzonadiol-4-yl)amino]-sn-glycerophosphocholine is inhibited by 75% at 5 mM 4-(2-aminoethyl)benzenesulfonyl fluoride
flippase activity for 1-oleoyl-2-[6-(7-nitrol-2-1,3-benzonadiol-4-yl)amino]-sn-glycerophosphoethanolamine is inhibited by 80% at 20 mM 5,5'-dithiobis(2-nitrobenzoic acid), flippase activity for 1-oleoyl-2-[6-(7-nitrol-2-1,3-benzonadiol-4-yl)amino]-sn-glycerophosphocholine is inhibited by 60% at 20 mM 5,5'-dithiobis(2-nitrobenzoic acid)
rat liver contains two populations, DEPC-sensitive and DEPC-insensitive, of flippases, which can be in a different of DEPC sensitivity or be two different proteins
transport of 0.001 mM tetramethylrosamine is essentially abolished by 1 mM methyl-beta-cyclodextrin, and transport of 0.005 mM H33342 is almost completely inhibited by 5 mM methyl-beta-cyclodextrin
prolonged treatment of erythrocytes with ribavirin results in surface exposure of phosphatidylserine, mainly caused by inactivation of the aminophospholipid translocase. Inactivation is due to severe ATP depletion
i.e. SNCEE, causes intracellular and extracellular trans-nitrosylation of proteins, respectively. Nitrosative stress inhibits the enzyme, and SNCEE causes significant S-nitrosylation/oxidation of thiols in HL-60 cells. SNCEE also strongly inhibites APLT, activated scramblase, and causes PS externalization, reversible by DTT
competitive inhibitor of ATP towards both Mg2+-ATPase activity and aminophospholipid translocation. Inhibition of translocation occurs at higher inhibitor concentration than the inhibition of Mg2+-ATPase activity
rat liver contains two populations of, NEM-sensitive and NEM-insensitive, flippases, which can be in a different of NEM sensitivity or be two different proteins
neither lipopolysaccharide from the Ra mutant of Escherichia coli nor deep rough chemotype lipopolysaccharide affect MsbA flippase activity significantly
neither lipopolysaccharide from the Ra mutant of Escherichia coli nor deep rough chemotype lipopolysaccharide affect MsbA flippase activity significantly
APLT is sensitive to redox modifications of its sulfhydryl groups, macrophages can directly participate in apoptotic cell clearance by S-nitrosylation/oxidation and inhibition of APLT causing PS externalization, reversible by DTT, overview, no inhibition and phagocytosis stimulation by S-nitrosoglutathione
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain
not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain; not inhibited by ouabain