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3.4.21.73: u-Plasminogen activator

This is an abbreviated version!
For detailed information about u-Plasminogen activator, go to the full flat file.

Word Map on EC 3.4.21.73

Reaction

Specific cleavage of Arg-/-Val bond in plasminogen to form plasmin =

Synonyms

Abbokinase, Cellular plasminogen activator, Double-chain urokinase-type plasminogen activator, EC 3.4.21.31, EC 3.4.99.26, Plasminogen activator, urokinase-type, PLAU, Two-chain urokinase-type plasminogen activator, u-PA, U-plasminogen activator, UK, uPA, uPA-type Plg activator, Urinary esterase A, Urinary plasminogen activator, Urokinase, Urokinase plasminogen activator, urokinase type plasminogen activator, urokinase-plasminogen activator, urokinase-type PA, urokinase-type plasmin activator, urokinase-type plasminogen, Urokinase-type plasminogen activator, urokinase-type Plg activator, urokine-type plasminogen activator

ECTree

     3 Hydrolases
         3.4 Acting on peptide bonds (peptidases)
             3.4.21 Serine endopeptidases
                3.4.21.73 u-Plasminogen activator

KM Value

KM Value on EC 3.4.21.73 - u-Plasminogen activator

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KM VALUE [mM]
SUBSTRATE
ORGANISM
UNIPROT
COMMENTARY hide
LITERATURE
IMAGE
0.052 - 0.6
GSGRSA
0.03 - 3.8
HYGRSA
0.297 - 0.608
L-diglutamyl-glycyl-L-arginine-4-nitroanilide
0.053 - 0.452
L-pyroGlu-Gly-L-Arg-4-nitroanilide
0.08
L-pyroGlu-Gly-L-Arg-p-NA
-
pH 8.8, 37°C
0.053
N-benzyloxycarbonyl-Gly-Gly-Arg-7-amido-4-trifluoromethylcoumarin
-
-
0.014 - 2.2
PFGRSA
0.000243 - 0.017
plasminogen
-
0.1 - 0.13
pyroGlu-Gly-Arg-4-nitroanilide
0.13 - 2.18
QRGRSA
0.051 - 0.089
S2444
0.13 - 2.3
YGAKAY
additional information
additional information
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