EC Number |
IC50 Value |
IC50 Value Maximum |
Inhibitor |
Reference |
---|
2.7.11.11 | 0.0000074 |
- |
cAMP-dependent protein kinase inhibitor(5-24) |
25°C, pH 7.4, wild-type enzyme |
761094 |
2.7.11.11 | 0.0000118 |
- |
rhodamine B-PKI(14-22)-GFMK |
pH and temperature not specified in the publication |
739224 |
2.7.11.11 | 0.0000479 |
- |
myr-PKI(14-22) |
pH and temperature not specified in the publication |
739224 |
2.7.11.11 | 0.0000606 |
- |
N-[2-(p-bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide |
25°C, pH 7.4, mutant enzyme L205R |
761094 |
2.7.11.11 | 0.0000633 |
- |
N-[2-(p-bromocinnamylamino)ethyl]-5-isoquinolinesulfonamide |
25°C, pH 7.4, wild-type enzyme |
761094 |
2.7.11.11 | 0.00187 |
- |
cAMP-dependent protein kinase inhibitor(5-24) |
25°C, pH 7.4, mutant enzyme L205R |
761094 |