Crystallization (Comment) | Organism |
---|---|
in complex with inhibitor biphenylacetyl-(Nepsilon-biphenylacetyl)-L-Lys-D-Arg-L-Tyr-N-phenylethyl, hanging drop vapor diffusion method, using 19%(w/v) polyethylene glycol 8000 and 200 mM ammonium sulfate, or in complex with inhibitor biphenylacetyl-(Nepsilon-biphenylacetyl)L-Lys-D-Arg-L-Phe-N-phenylethyl hanging drop vapor diffusion method, using 25% (w/v) polyethylene glycol 8000 and 200 mM ammonium sulfate, or in complex with biphenylacetyl-M-Cys-D-Arg-L-Phe-N-phenylethyl, hanging drop vapor diffusion method, using 30% (w/v) polyethylene glycol 8000 and 200 mM ammonium sulfate | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
biphenylacetyl-(N6-biphenylacetyl)-Lys-D-Arg-Tyr-N-phenylethyl | - |
Homo sapiens | |
biphenylacetyl-(N6-biphenylacetyl)Lys-D-Arg-Phe-N-phenylethyl | - |
Homo sapiens | |
biphenylacetyl-MCys-D-Arg-Phe-N-phenylethyl | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P07711 | - |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.000019 | - |
biphenylacetyl-MCys-D-Arg-Phe-N-phenylethyl | pH and temperature not specified in the publication | Homo sapiens | |
0.000023 | - |
biphenylacetyl-(N6-biphenylacetyl)-Lys-D-Arg-Tyr-N-phenylethyl | pH and temperature not specified in the publication | Homo sapiens | |
0.000511 | - |
biphenylacetyl-(N6-biphenylacetyl)Lys-D-Arg-Phe-N-phenylethyl | pH and temperature not specified in the publication | Homo sapiens |