Inhibitors | Comment | Organism | Structure |
---|---|---|---|
4-amidinophenylpyruvate | - |
Homo sapiens | |
benzamidine | - |
Homo sapiens | |
additional information | computational modeling, inhibitor binding mechanism, preference of binding of different benzamidine derivatives due to thermodynamic measurements and and hydration in descending order: 4-(2-oxo-1-propyl)benzamidine, 4-ethylbenzamidine, 4-(1-propyl)benzamidine, 4-methylbenzamidine, benzamidine, 4-amidinophenylpyruvate, inhibitors bind to Ser195 | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P00734 | - |
- |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0003 | - |
benzamidine | - |
Homo sapiens | |
0.00062 | - |
4-amidinophenylpyruvate | - |
Homo sapiens |