Inhibitors | Comment | Organism | Structure |
---|---|---|---|
L-MetStaCys | - |
Escherichia coli | |
L-MetStaCys | - |
Pyrococcus furiosus | |
L-MetStaVal | - |
Escherichia coli | |
L-MetStaVal | - |
Pyrococcus furiosus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.59 | - |
L-Met-p-nitroanilide | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Pyrococcus furiosus | |
3 | - |
L-Met-p-nitroanilide | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Escherichia coli | |
5.1 | - |
Met-Gly-Met-Met | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Pyrococcus furiosus | |
18.3 | - |
Met-Gly-Met-Met | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Escherichia coli |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Escherichia coli | - |
- |
- |
Pyrococcus furiosus | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
L-Met-p-nitroanilide + H2O | - |
Escherichia coli | p-nitroaniline + L-Met | - |
? | |
L-Met-p-nitroanilide + H2O | - |
Pyrococcus furiosus | p-nitroaniline + L-Met | - |
? | |
Met-Gly-Met-Met + H2O | - |
Escherichia coli | Gly-Met-Met + Met | - |
? | |
Met-Gly-Met-Met + H2O | - |
Pyrococcus furiosus | Gly-Met-Met + Met | - |
? |
Synonyms | Comment | Organism |
---|---|---|
MetAP-I | - |
Escherichia coli |
MetAP-II | - |
Pyrococcus furiosus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.006 | - |
L-Met-p-nitroanilide | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Escherichia coli | |
0.057 | - |
L-Met-p-nitroanilide | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Pyrococcus furiosus | |
18.3 | - |
Met-Gly-Met-Met | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Escherichia coli | |
188 | - |
Met-Gly-Met-Met | in 25 mM HEPES buffer at 30°C (pH 7.5) with 150 mM KCl | Pyrococcus furiosus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0017 | - |
in 25 mM HEPES buffer at 30°C (pH 7.5) | Pyrococcus furiosus | L-MetStaCys | |
0.002 | - |
in 25 mM HEPES buffer at 30°C (pH 7.5) | Pyrococcus furiosus | L-MetStaVal | |
0.0025 | - |
in 25 mM HEPES buffer at 30°C (pH 7.5) | Escherichia coli | L-MetStaCys | |
0.0043 | - |
in 25 mM HEPES buffer at 30°C (pH 7.5) | Escherichia coli | L-MetStaVal |