Cloned (Comment) | Organism |
---|---|
Epac1-camps-PDE3A fusion protein is expressed in HEK-293 cells | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Cilostamide | - |
Homo sapiens | |
IBMX | - |
Homo sapiens | |
Milrinone | - |
Homo sapiens | |
additional information | not inhibited by rolipram and sildenafil | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P27815 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
3',5'-cAMP + H2O | - |
Homo sapiens | 5'-AMP | - |
? | |
3',5'-cGMP + H2O | - |
Homo sapiens | 5'-GMP | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PDE3 | - |
Homo sapiens |
PDE3A | isoform | Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00037 | - |
- |
Homo sapiens | Cilostamide | |
0.007 | - |
- |
Homo sapiens | Milrinone | |
0.0127 | - |
- |
Homo sapiens | IBMX |