Inhibitors | Comment | Organism | Structure |
---|---|---|---|
apigenin | IC50: 0.0105 mM, PDB3; IC50: 0.0167 mM, PDB2; IC50: 0.0254 mM, PDB1 | Cavia porcellus | |
Biochanin A | IC50: 0.0279 mM, PDE2; IC50: 0.0291 mM, PDE1 | Cavia porcellus | |
daidzein | IC50: 0.0286 mM, PDE3 | Cavia porcellus | |
diosmetin | IC50: 0.0048 mM, PDB2; IC50: 0.0144 mM, PDB1 | Cavia porcellus | |
eriodictyol | IC50: 0.0525 mM, PDB3 | Cavia porcellus | |
genistein | IC50: 0.0017 mM, PDB2; IC50: 0.0129 mM, PDB3; IC50: 0.0168 mM, PDB1 | Cavia porcellus | |
luteolin | IC50: 0.0101 mM, PDB3; IC50: 0.0133 mM, PDB2; IC50: 0.0215 mM, PDB1 | Cavia porcellus | |
luteolin-7-glucoside | IC50: 0.0351 mM, PDB2 | Cavia porcellus | |
myricetin | IC50: 0.0124 mM, PDB3; IC50: 0.0128 mM, PDB2; IC50: 0.0249 mM, PDB1 | Cavia porcellus | |
quercetin | IC50: 0.0056 mM, PDB3; IC50: 0.0179 mM, PDB2; IC50: 0.0278 mM, PDB1 | Cavia porcellus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Cavia porcellus | - |
- |
- |
Synonyms | Comment | Organism |
---|---|---|
PDB1 | - |
Cavia porcellus |
PDB2 | - |
Cavia porcellus |
PDB3 | - |
Cavia porcellus |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0017 | - |
IC50: 0.0017 mM, PDB2 | Cavia porcellus | genistein | |
0.0048 | - |
IC50: 0.0048 mM, PDB2 | Cavia porcellus | diosmetin | |
0.0056 | - |
IC50: 0.0056 mM, PDB3 | Cavia porcellus | quercetin | |
0.0101 | - |
IC50: 0.0101 mM, PDB3 | Cavia porcellus | luteolin | |
0.0105 | - |
IC50: 0.0105 mM, PDB3 | Cavia porcellus | apigenin | |
0.0124 | - |
IC50: 0.0124 mM, PDB3 | Cavia porcellus | myricetin | |
0.0128 | - |
IC50: 0.0128 mM, PDB2 | Cavia porcellus | myricetin | |
0.0129 | - |
IC50: 0.0129 mM, PDB3 | Cavia porcellus | genistein | |
0.0133 | - |
IC50: 0.0133 mM, PDB2 | Cavia porcellus | luteolin | |
0.0144 | - |
IC50: 0.0144 mM, PDB1 | Cavia porcellus | diosmetin | |
0.0167 | - |
IC50: 0.0167 mM, PDB2 | Cavia porcellus | apigenin | |
0.0168 | - |
IC50: 0.0168 mM, PDB1 | Cavia porcellus | genistein | |
0.0179 | - |
IC50: 0.0179 mM, PDB2 | Cavia porcellus | quercetin | |
0.0215 | - |
IC50: 0.0215 mM, PDB1 | Cavia porcellus | luteolin | |
0.0249 | - |
IC50: 0.0249 mM, PDB1 | Cavia porcellus | myricetin | |
0.0254 | - |
IC50: 0.0254 mM, PDB1 | Cavia porcellus | apigenin | |
0.0278 | - |
IC50: 0.0278 mM, PDB1 | Cavia porcellus | quercetin | |
0.0279 | - |
IC50: 0.0279 mM, PDE2 | Cavia porcellus | Biochanin A | |
0.0286 | - |
IC50: 0.0286 mM, PDE3 | Cavia porcellus | daidzein | |
0.0291 | - |
IC50: 0.0291 mM, PDE1 | Cavia porcellus | Biochanin A | |
0.0351 | - |
IC50: 0.0351 mM, PDB2 | Cavia porcellus | luteolin-7-glucoside | |
0.0525 | - |
IC50: 0.0525 mM, PDB3 | Cavia porcellus | eriodictyol |