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Literature summary for 3.1.1.8 extracted from

  • Al-Aboudi, A.; Odeh, H.; Khalid, A.; Naz, Q.; Choudhary, M.I.
    Butyrylcholinesterase inhibitory activity of testosterone and some of its metabolites (2008), J. Enzyme Inhib. Med. Chem., 24, 553-558.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
1-dehydrotestosterone
-
Equus caballus
11alpha,17beta-dihydroxyandrost-1,4-dien-3-one
-
Equus caballus
11alpha-hydroxyandrost-1,4-dien-3,17-dione
-
Equus caballus
11alpha-hydroxyandrost-4-en-3,17-dione
-
Equus caballus
11alpha-hydroxytestolactone
-
Equus caballus
11alpha-hydroxytestosterone
-
Equus caballus
17beta-hydroxy-5alpha-androstan-3,6-dione
-
Equus caballus
androst-1,4-dien-3,17-dione
-
Equus caballus
androst-4-en-3,7-dione
-
Equus caballus
galanthamine
-
Equus caballus
additional information molecular docking analysis of inhibitors, overview Equus caballus
testolactone
-
Equus caballus
testosterone
-
Equus caballus

Localization

Localization Comment Organism GeneOntology No. Textmining
extracellular
-
Equus caballus
-
-

Organism

Organism UniProt Comment Textmining
Equus caballus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
serum
-
Equus caballus
-

Synonyms

Synonyms Comment Organism
BChE
-
Equus caballus
butyrylcholinesterase
-
Equus caballus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
additional information
-
additional information inhibition kinetics Equus caballus

IC50 Value

IC50 Value IC50 Value Maximum Comment Organism Inhibitor Structure
0.00155
-
-
Equus caballus androst-4-en-3,7-dione
0.0085
-
-
Equus caballus galanthamine
0.0209
-
-
Equus caballus 1-dehydrotestosterone
0.0535
-
-
Equus caballus testosterone
0.0615
-
-
Equus caballus 11alpha,17beta-dihydroxyandrost-1,4-dien-3-one
0.089
-
-
Equus caballus 11alpha-hydroxytestosterone
0.0959
-
-
Equus caballus 17beta-hydroxy-5alpha-androstan-3,6-dione
0.1027
-
-
Equus caballus androst-1,4-dien-3,17-dione
0.1413
-
-
Equus caballus 11alpha-hydroxyandrost-4-en-3,17-dione
0.1425
-
-
Equus caballus testolactone
0.1647
-
-
Equus caballus 11alpha-hydroxyandrost-1,4-dien-3,17-dione
0.284
-
-
Equus caballus 11alpha-hydroxytestolactone