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Literature summary for 3.1.1.8 extracted from

  • Bajgar, J.; Bartosova, L.; Kuca, K.; Jun, D.; Fusek, J.
    Changes of cholinesterase activities in the rat blood and brain after sarin intoxication pretreated with butyrylcholinesterase (2007), Drug Chem. Toxicol., 30, 351-359.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
additional information rat plasma BuChE is increased when pretreated with horse BuChE Rattus norvegicus

Inhibitors

Inhibitors Comment Organism Structure
sarin
-
Equus caballus

Localization

Localization Comment Organism GeneOntology No. Textmining
extracellular
-
Rattus norvegicus
-
-
extracellular
-
Equus caballus
-
-

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
butyrylthiocholine + H2O Rattus norvegicus
-
thiocholine + butyrate
-
?
butyrylthiocholine + H2O Equus caballus
-
thiocholine + butyrate
-
?
additional information Equus caballus rat plasma BuChE is increased when pretreated with horse BuChE ?
-
?

Organism

Organism UniProt Comment Textmining
Equus caballus
-
-
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
blood plasma
-
Rattus norvegicus
-
blood plasma
-
Equus caballus
-

Specific Activity [micromol/min/mg]

Specific Activity Minimum [µmol/min/mg] Specific Activity Maximum [µmol/min/mg] Comment Organism
additional information
-
plasma BuChE before and after sarin inhalation exposure of untreated rats and animals pretreated with horse BuChE Rattus norvegicus
additional information
-
plasma BuChE before and after sarin inhalation exposure of untreated rats and animals pretreated with horse BuChE Equus caballus

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
butyrylthiocholine + H2O
-
Rattus norvegicus thiocholine + butyrate
-
?
butyrylthiocholine + H2O
-
Equus caballus thiocholine + butyrate
-
?
additional information rat plasma BuChE is increased when pretreated with horse BuChE Equus caballus ?
-
?

Synonyms

Synonyms Comment Organism
BuChE
-
Rattus norvegicus
butyrylcholinesterase
-
Rattus norvegicus
butyrylcholinesterase
-
Equus caballus
EqBuChE
-
Equus caballus