Inhibitors | Comment | Organism | Structure |
---|---|---|---|
benzoylthiocholine | substrate inhibition | Rattus norvegicus | |
Triton X-100 | inhibition above 0.01 mM | Rattus norvegicus |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.047 | - |
Benzoylcholine | pH 7.4, 37°C | Rattus norvegicus | |
0.06 | - |
acetylthiocholine | pH 7.4, 37°C | Rattus norvegicus | |
0.087 | - |
acetylthiocholine | pH 7.4, 37°C | Rattus norvegicus | |
0.115 | - |
propionylthiocholine | pH 7.4, 37°C | Rattus norvegicus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Rattus norvegicus | - |
- |
- |
Purification (Comment) | Organism |
---|---|
260fold | Rattus norvegicus |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
intestine | - |
Rattus norvegicus | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
4612 | - |
- |
Rattus norvegicus |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
acetylthiocholine + H2O | increasing activity with substrates in the following order: acetylthiocholine, propionylthiocholine, butyrylthiocholine | Rattus norvegicus | thiocholine + acetate | - |
? | |
benzoylcholine + H2O | - |
Rattus norvegicus | choline + benzoate | - |
? | |
butyrylthiocholine + H2O | increasing activity with substrates in the following order: acetylthiocholine, propionylthiocholine, butyrylthiocholine | Rattus norvegicus | thiocholine + butyrate | - |
? | |
propionylthiocholine + H2O | increasing activity with substrates in the following order: acetylthiocholine, propionylthiocholine, butyrylthiocholine | Rattus norvegicus | thiocholine + propionate | - |
? |
Subunits | Comment | Organism |
---|---|---|
tetramer | nonreducing PAGE | Rattus norvegicus |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
- |
Rattus norvegicus |
Turnover Number Minimum [1/s] | Turnover Number Maximum [1/s] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.005 | - |
acetylthiocholine | pH 7.4, 37°C | Rattus norvegicus | |
16.8 | - |
Benzoylcholine | pH 7.4, 37°C | Rattus norvegicus | |
23.5 | - |
acetylthiocholine | pH 7.4, 37°C | Rattus norvegicus | |
49.2 | - |
propionylthiocholine | pH 7.4, 37°C | Rattus norvegicus |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.2 | - |
- |
Rattus norvegicus |