Crystallization (Comment) | Organism |
---|---|
phospholipase A2 complexed with berberine, hanging drop vapor diffusion method, using 5 mM CaCl2 in 25 mM sodium acetate buffer of pH 6.2 with 15% (w/v) polyethylene glycol 8000 and 0.2 M ammonium sulfate | Daboia russelii russelii |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
ajmaline | - |
Daboia russelii russelii | |
Anisic acid | - |
Daboia russelii russelii | |
aristolochic acid | - |
Daboia russelii russelii | |
Berberine | competitive inhibitor of phospholipase A2 | Daboia russelii russelii | |
diclofenac | - |
Daboia russelii russelii | |
oxyphenbutazone | - |
Daboia russelii russelii |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.02 | - |
soya lecithin | at pH 8.9, temperature not specified in the publication | Daboia russelii russelii |
Natural Substrates | Organism | Comment (Nat. Sub.) | Natural Products | Comment (Nat. Pro.) | Rev. | Reac. |
---|---|---|---|---|---|---|
soya lecithin + H2O | Daboia russelii russelii | - |
? | - |
? |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Daboia russelii russelii | P59071 | Indian Russell's viper, chain viper | - |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
venom | - |
Daboia russelii russelii | - |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
soya lecithin + H2O | - |
Daboia russelii russelii | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
PLA2 | - |
Daboia russelii russelii |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.021 | - |
Berberine | at pH 8.9, temperature not specified in the publication | Daboia russelii russelii |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.087 | - |
at pH 8.9, temperature not specified in the publication | Daboia russelii russelii | Berberine |