Activating Compound | Comment | Organism | Structure |
---|---|---|---|
pioglitazone | a thiazolidinedione, activates PI3K 2-2.5fold at 0.002-0.010 mM, activates adiponectin secretion from adipocytes in vivo | Mus musculus | |
pioglitazone | a thiazolidinedione, activates PI3K 2-2.5fold at 0.002-0.010 mM, activates adiponectin secretion from adipocytes in vivo | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
Wortmannin | - |
Homo sapiens | |
Wortmannin | - |
Mus musculus |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Mus musculus | - |
- |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
3T3-L1 cell | - |
Mus musculus | - |
adipocyte | - |
Mus musculus | - |
adipocyte | primary, obtained from subcutaneous tissue biopsies performed on two lean non-diabetic male subjects | Homo sapiens | - |
cell culture | - |
Mus musculus | - |
fibroblast | - |
Mus musculus | - |
Synonyms | Comment | Organism |
---|---|---|
PI3K | - |
Mus musculus |
PI3K | - |
Homo sapiens |
General Information | Comment | Organism |
---|---|---|
physiological function | the thiazolidinedione pioglitazone acutely stimulates adiponectin secretion from mouse and human adipocytes via activation of the phosphatidylinositol 3-kinase | Mus musculus |
physiological function | the thiazolidinedione pioglitazone acutely stimulates adiponectin secretion from mouse and human adipocytes via activation of the phosphatidylinositol 3-kinase | Homo sapiens |