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Literature summary for 2.7.1.137 extracted from

  • Pereira, R.I.; Leitner, J.W.; Erickson, C.; Draznin, B.
    Pioglitazone acutely stimulates adiponectin secretion from mouse and human adipocytes via activation of the phosphatidylinositol 3-kinase (2008), Life Sci., 83, 638-643.
    View publication on PubMed

Activating Compound

Activating Compound Comment Organism Structure
pioglitazone a thiazolidinedione, activates PI3K 2-2.5fold at 0.002-0.010 mM, activates adiponectin secretion from adipocytes in vivo Mus musculus
pioglitazone a thiazolidinedione, activates PI3K 2-2.5fold at 0.002-0.010 mM, activates adiponectin secretion from adipocytes in vivo Homo sapiens

Inhibitors

Inhibitors Comment Organism Structure
Wortmannin
-
Homo sapiens
Wortmannin
-
Mus musculus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Mus musculus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
3T3-L1 cell
-
Mus musculus
-
adipocyte
-
Mus musculus
-
adipocyte primary, obtained from subcutaneous tissue biopsies performed on two lean non-diabetic male subjects Homo sapiens
-
cell culture
-
Mus musculus
-
fibroblast
-
Mus musculus
-

Synonyms

Synonyms Comment Organism
PI3K
-
Mus musculus
PI3K
-
Homo sapiens

General Information

General Information Comment Organism
physiological function the thiazolidinedione pioglitazone acutely stimulates adiponectin secretion from mouse and human adipocytes via activation of the phosphatidylinositol 3-kinase Mus musculus
physiological function the thiazolidinedione pioglitazone acutely stimulates adiponectin secretion from mouse and human adipocytes via activation of the phosphatidylinositol 3-kinase Homo sapiens