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Literature summary for 2.5.1.15 extracted from

  • Williams, D.L.; Spring, L.; Harris, E.; Roche, P.; Gillis, T.P.
    Dihydropteroate synthase of Mycobacterium leprae and dapsone resistance (2000), Antimicrob. Agents Chemother., 44, 1530-1537.
    View publication on PubMedView publication on EuropePMC

Cloned(Commentary)

Cloned (Comment) Organism
expression in Escherichia coli C600 and in Escherichia coli folP knockout mutant Mycobacterium leprae

Inhibitors

Inhibitors Comment Organism Structure
dapsone
-
Mycobacterium leprae

KM Value [mM]

KM Value [mM] KM Value Maximum [mM] Substrate Comment Organism Structure
additional information
-
additional information activity in Escherichia coli C600 and recombinant strains Mycobacterium leprae

Natural Substrates/ Products (Substrates)

Natural Substrates Organism Comment (Nat. Sub.) Natural Products Comment (Nat. Pro.) Rev. Reac.
2-amino-4-hydroxy-6-hydroxymethyl-7,8-dihydropteridine diphosphate + 4-aminobenzoate Mycobacterium leprae
-
diphosphate + 7,8-dihydropteroate
-
?

Organism

Organism UniProt Comment Textmining
Mycobacterium leprae P0C0X1
-
-
Mycobacterium leprae P0C0X2
-
-

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
2-amino-4-hydroxy-6-hydroxymethyl-7,8-dihydropteridine diphosphate + 4-aminobenzoate
-
Mycobacterium leprae diphosphate + 7,8-dihydropteroate
-
?