KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
additional information | - |
additional information | kinetics | Homo sapiens | |
4.9 | - |
serotonin | lung UGT1A6, pH 7.5, 37°C | Homo sapiens | |
5.2 | 8.8 | serotonin | liver UGT1A6, pH 7.5, 37°C | Homo sapiens | |
6.5 | - |
serotonin | kidney UGT1A6, pH 7.5, 37°C | Homo sapiens | |
12.4 | - |
serotonin | intestine UGT1A6, pH 7.5, 37°C | Homo sapiens | |
55.9 | - |
serotonin | recombinant UGT1A6 from lymphoblasts or insect cells, pH 7.5, 37°C | Homo sapiens |
Localization | Comment | Organism | GeneOntology No. | Textmining |
---|---|---|---|---|
microsome | - |
Homo sapiens | - |
- |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | P19224 | - |
- |
Source Tissue | Comment | Organism | Textmining |
---|---|---|---|
intestine | - |
Homo sapiens | - |
kidney | - |
Homo sapiens | - |
liver | - |
Homo sapiens | - |
lung | - |
Homo sapiens | - |
additional information | tissue-specific serotonin glucuronidation activity | Homo sapiens | - |
Specific Activity Minimum [µmol/min/mg] | Specific Activity Maximum [µmol/min/mg] | Comment | Organism |
---|---|---|---|
additional information | - |
activity of isozyme UGT1A6 in microsomes of different tissues | Homo sapiens |
0.00077 | 0.033 | liver UGT1A6 of different individuals, microsomes | Homo sapiens |
0.0158 | - |
recombinant UGT1A6 from lymphoblasts or insect cells, microsomes | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
UDP-glucuronate + 4-nitrophenol | recombinant isozyme UGT1A6 from lymphoblasts or insect cells | Homo sapiens | UDP + 4-nitrophenyl beta-D-glucuronide | - |
? | |
UDP-glucuronate + serotonin | in vitro substrate, isozyme UGT1A6 | Homo sapiens | UDP + serotonin beta-D-glucuronide | - |
? |
Synonyms | Comment | Organism |
---|---|---|
UDP-glucuronosyltransferase 1A6 | - |
Homo sapiens |
UGT1A6 | - |
Homo sapiens |
Temperature Optimum [°C] | Temperature Optimum Maximum [°C] | Comment | Organism |
---|---|---|---|
37 | - |
assay at | Homo sapiens |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | - |
assay at | Homo sapiens |