Cloned (Comment) | Organism |
---|---|
expressed in Baculovirus Bac-N-Blue expression system | Homo sapiens |
Inhibitors | Comment | Organism | Structure |
---|---|---|---|
BMS-303141 | - |
Homo sapiens | |
Hydroxycitrate | competitive | Homo sapiens | |
SB-201076 | - |
Homo sapiens |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.004 | - |
CoA | direct assay | Homo sapiens | |
0.014 | - |
CoA | coupled assay | Homo sapiens | |
0.047 | - |
ATP | direct assay | Homo sapiens | |
0.0738 | - |
citrate | direct assay | Homo sapiens | |
0.098 | - |
citrate | coupled assay | Homo sapiens | |
0.12 | - |
ATP | coupled assay | Homo sapiens |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | - |
Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | - |
- |
- |
Purification (Comment) | Organism |
---|---|
ammonium sulfate precipitation, ion exchange chromatography (DEAE), gel filtration | Homo sapiens |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
citrate + CoA + ATP | - |
Homo sapiens | acetyl-CoA + oxaloacetate + ADP + phosphate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
ATP citrate lyase | - |
Homo sapiens |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.00015 | - |
Hydroxycitrate | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.00094 | - |
- |
Homo sapiens | BMS-303141 |