Inhibitors | Comment | Organism | Structure |
---|---|---|---|
betulin | IC50: 0.083 mM, hACAT-1 | Homo sapiens | |
lupeol | IC50: 0.048 mM, hACAT-1 | Homo sapiens |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Homo sapiens | O75908 | - |
- |
Homo sapiens | P35610 | - |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
oleoyl-CoA + cholesterol | - |
Homo sapiens | CoA + cholesteryl oleate | - |
? |
Synonyms | Comment | Organism |
---|---|---|
hACAT-1 | - |
Homo sapiens |
hACAT-2 | - |
Homo sapiens |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.048 | - |
IC50: 0.048 mM, hACAT-1 | Homo sapiens | lupeol | |
0.083 | - |
IC50: 0.083 mM, hACAT-1 | Homo sapiens | betulin |