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Literature summary for 2.1.1.8 extracted from

  • Taraschenko, O.D.; Barnes, W.G.; Herrick-Davis, K.; Yokoyama, Y.; Boyd, D.L.; Hough, L.B.
    Actions of tacrine and galanthamine on histamine-N-methyltransferase (2005), Methods Find. Exp. Clin. Pharmacol., 27, 161-165.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
additional information not inhibitory: galanthamine up to 0.001 mM Homo sapiens
additional information not inhibitory: galanthamine up to 0.001 mM Rattus norvegicus
tacrine 50% inhibition at 0.00046 mM for enzyme of embryonic kidney, at 0.0007 mM for recombinant brain enzyme Homo sapiens
tacrine 50% inhibition at 0.00029 mM Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Homo sapiens
-
-
-
Rattus norvegicus
-
-
-

Source Tissue

Source Tissue Comment Organism Textmining
brain recombinant enzyme from brain Homo sapiens
-
kidney
-
Rattus norvegicus
-
kidney embryonic cells Homo sapiens
-