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Literature summary for 1.4.3.4 extracted from

  • Osman, M.Y.; Osman, H.M.
    Inhibitory effect of acetylcholine on monoamine oxidase A and B activity in different parts of rat brain (2008), Arzneimittelforschung, 58, 493-496.
    View publication on PubMed

Inhibitors

Inhibitors Comment Organism Structure
Acetylcholine competitively inhibits monoamine oxidase A in the brain in a tissue-dependent manner, inhibition of MAO-A in cerebellum; competitively inhibits monoamine oxidase B in the brain in a tissue-dependent manner, inhibition of MAO-B in basal ganglia Rattus norvegicus

Organism

Organism UniProt Comment Textmining
Rattus norvegicus P19643 MAO-B; male albino rats, isozyme MAO-B
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Rattus norvegicus P21396 MAO-A; male albino rats, isozyme MAO-A
-

Source Tissue

Source Tissue Comment Organism Textmining
brain
-
Rattus norvegicus
-

Synonyms

Synonyms Comment Organism
MAO-A
-
Rattus norvegicus
MAO-B
-
Rattus norvegicus
monoamine oxidase A
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Rattus norvegicus
monoamine oxidase B
-
Rattus norvegicus

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
additional information
-
additional information values for inhibition of isozyme MAO-A by acetylcholine are higher than those for isozyme MAO-B Rattus norvegicus