Inhibitors | Comment | Organism | Structure |
---|---|---|---|
dehydroluciferyl-adenylate | tight-binding competitive inhibitor | Photinus pyralis | |
oxyluciferin | competitive inhibitor | Photinus pyralis |
KM Value [mM] | KM Value Maximum [mM] | Substrate | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0147 | - |
oxyluciferin | - |
Photinus pyralis | |
0.0149 | - |
dehydroluciferyl-adenylate | - |
Photinus pyralis |
Metals/Ions | Comment | Organism | Structure |
---|---|---|---|
Mg2+ | required | Photinus pyralis |
Organism | UniProt | Comment | Textmining |
---|---|---|---|
Photinus pyralis | - |
- |
- |
Substrates | Comment Substrates | Organism | Products | Comment (Products) | Rev. | Reac. |
---|---|---|---|---|---|---|
ATP + O2 + oxyluciferin | assay at pH 7.5, 24-27°C | Photinus pyralis | ? | - |
? | |
D-luciferin + ATP + O2 | assay at pH 7.5, 24-27°C | Photinus pyralis | ? | - |
? |
Synonyms | Comment | Organism |
---|---|---|
firefly luciferase | - |
Photinus pyralis |
Luc | - |
Photinus pyralis |
Temperature Minimum [°C] | Temperature Maximum [°C] | Comment | Organism |
---|---|---|---|
24 | 27 | assay at | Photinus pyralis |
pH Optimum Minimum | pH Optimum Maximum | Comment | Organism |
---|---|---|---|
7.5 | - |
assay at | Photinus pyralis |
Ki Value [mM] | Ki Value maximum [mM] | Inhibitor | Comment | Organism | Structure |
---|---|---|---|---|---|
0.0000038 | - |
dehydroluciferyl-adenylate | - |
Photinus pyralis | |
0.0005 | - |
oxyluciferin | - |
Photinus pyralis |
IC50 Value | IC50 Value Maximum | Comment | Organism | Inhibitor | Structure |
---|---|---|---|---|---|
0.0000074 | - |
2.5 nM D-luciferin | Photinus pyralis | dehydroluciferyl-adenylate | |
0.0000085 | - |
5 nM D-luciferin | Photinus pyralis | dehydroluciferyl-adenylate | |
0.0000103 | - |
10 nM D-luciferin | Photinus pyralis | dehydroluciferyl-adenylate | |
0.0000132 | - |
20 nM D-luciferin | Photinus pyralis | dehydroluciferyl-adenylate | |
0.000022 | - |
40 nM D-luciferin | Photinus pyralis | dehydroluciferyl-adenylate |