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Literature summary for 1.13.12.5 extracted from

  • Auld, D.S.; Thorne, N.; Maguire, W.F.; Inglese, J.
    Mechanism of PTC124 activity in cell-based luciferase assay of nonsense codon suppression (2009), Proc. Natl. Acad. Sci. USA, 106, 3585-3590.
    View publication on PubMedView publication on EuropePMC

Activating Compound

Activating Compound Comment Organism Structure
MS-275
-
Renilla reniformis

Cloned(Commentary)

Cloned (Comment) Organism
expression in HEK-293 cells or Grip-Tite 293 MSR cells Renilla reniformis

Protein Variants

Protein Variants Comment Organism
T329G no significant influence on enzyme activity Renilla reniformis

Inhibitors

Inhibitors Comment Organism Structure
N-benzyl-4-methylbenzenesulfonamide inhibition of purified enzyme, inducing activity in cell-based assay Renilla reniformis

Organism

Organism UniProt Comment Textmining
Renilla reniformis
-
-
-

Purification (Commentary)

Purification (Comment) Organism
-
Renilla reniformis

Substrates and Products (Substrate)

Substrates Comment Substrates Organism Products Comment (Products) Rev. Reac.
coelenterazine-H + O2 5 microM, assay at pH 7.5 Renilla reniformis ?
-
?

Synonyms

Synonyms Comment Organism
Renilla reniformis luciferase
-
Renilla reniformis
RLuc
-
Renilla reniformis

pH Optimum

pH Optimum Minimum pH Optimum Maximum Comment Organism
7.5
-
assay at Renilla reniformis

Ki Value [mM]

Ki Value [mM] Ki Value maximum [mM] Inhibitor Comment Organism Structure
0.0012
-
N-benzyl-4-methylbenzenesulfonamide
-
Renilla reniformis