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0.0443
(2alpha,3beta)-2,3-dihydroxyurs-12-en-28-oic acid
Rattus norvegicus
-
IC50: 0.0443 mM
0.0098
(2E)-1-[2,4-dihydroxy-6-methoxy-3-[(2R)-5-methyl-2-(1-methylethenyl)hex-4-en-1-yl]phenyl]-3-(2,4-dihydroxyphenyl)prop-2-en-1-one
Rattus norvegicus
-
IC50: 0.0098 mM
0.0298
(2E,4Z,8E)-N-[9-(3,4-methylenedioxyphenyl)-2,4,8-nonatrienoyl]piperidine
Rattus norvegicus
-
IC50: 0.0298 mM, isolated from the extracts of fruits of Piper longum and Piper nigrum
0.01
(2S)-1-(3-[[(2S)-1-ethoxy-4-phenylbutan-2-yl]sulfamoyl]anilino)-4-methyl-1-oxopentan-2-yl 2,2-dimethylpropanoate
Homo sapiens
-
IC50 less than 0.01 mM, at pH 7.5 and 25°C
0.000011
(2S)-1-[(1-[[(1S)-1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-3-phenylpropyl]carbamoyl]cyclopentyl)amino]-4-methyl-1-oxopentan-2-yl 2,2-dimethylpropanoate
Homo sapiens
-
at pH 7.5 and 25°C
0.000326
(4-[4-[4-(2-amino-5-chlorobenzamido)phenyl]thieno[3,2-d]pyrimidin-7-yl]cyclohexyl)acetic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
0.000276
(4-[4-[4-(3-chlorobenzamido)phenyl]thieno[3,2-d]pyrimidin-7-yl]cyclohexyl)acetic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
0.001
(4-[4-[4-(5-chloro-2-nitrobenzamido)phenyl]thieno[3,2-d]pyrimidin-7-yl]cyclohexyl)acetic acid
Homo sapiens
above, pH 7.4, 25°C
0.000351
(4-[4-[4-([[2-fluoro-5-(trifluoromethyl)phenyl]carbamoyl]amino)phenyl]thieno[3,2-d]pyrimidin-7-yl]cyclohexyl)acetic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
0.00046
(4S,7R)-4-(5,5-dimethyl-4-oxo-4,5-dihydrofuran-2-yl)-2,2-dimethyl-4,7-bis[(4E)-4-methyl-5-[(2R)-4-methyl-6-oxo-3,6-dihydro-2H-pyran-2-yl]pent-4-en-1-yl]-4,5,6,7-tetrahydro-1-benzofuran-3(2H)-one
Homo sapiens
pH 7.4, temperature not specified in the publication
0.00036
(trans-4-(4-[(5-benzyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl)cyclohexyl)acetic acid
Homo sapiens
-
pH not specified in the publication, 25°C
0.000019
(trans-4-(4-[(5-cyclopentylethyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl)cyclohexyl)acetic acid
Homo sapiens
-
pH not specified in the publication, 25°C
0.000024
(trans-4-(4-[(5-cyclopentylmethyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl)cyclohexyl)acetic acid
Homo sapiens
-
pH not specified in the publication, 25°C
0.000045
(trans-4-(4-[(5-[1-fluorobenzyl]-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl)cyclohexyl)acetic acid
Homo sapiens
-
pH not specified in the publication, 25°C
0.00003
(trans-4-(4-[(5-[2-chlorobenzyl]-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl)cyclohexyl)acetic acid
Homo sapiens
-
pH not specified in the publication, 25°C
0.00003
(trans-4-(4-[(5-[2-fluorobenzyl]-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl)cyclohexyl)acetic acid
Homo sapiens
-
pH not specified in the publication, 25°C
0.000253
(trans-4-[4-[(3-benzyl-1,2,4-oxadiazol-5-yl)carbamoyl]phenyl]cyclohexyl)acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000286
(trans-4-[4-[(5-benzyl-1,2,4-oxadiazol-3-yl)carbamoyl]phenyl]cyclohexyl)acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000036
(trans-4-[4-[(5-benzyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenyl]cyclohexyl)acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000409
3-(4-[4-[4-(3-chlorobenzamido)phenyl]thieno[3,2-d]pyrimidin-7-yl]cyclohexyl)propanoic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
0.001
4-[4-[4-(3-chlorobenzamido)phenyl]thieno[3,2-d]pyrimidin-7-yl]cyclohexane-1-carboxylic acid
Homo sapiens
above, pH 7.4, 25°C
0.047 - 0.1607
7beta-(3-ethyl-cis-crotonoyloxy)-1alpha-(2-methylbutyryloxy)-3,14-dehydro-Z-notonipetranone
0.211 - 0.2944
8-angeloyloxy-3,4-epoxy-bisabola-7(14),10-dien-2-one
0.2
amidepsine C
Homo sapiens
-
-
0.0096
betulinic acid
Rattus norvegicus
-
a lupane-type triterpenoid, isolated from methanolic extracts of Alnus hirsuta, noncompetitive inhibition, IC50: 0.0096 mM
0.25
brachynereolide
Rattus norvegicus
-
IC50: 0.25 mM, above
0.000022
cis-4-(4-[[5-(cyclopentylamino)-1,3,4-thiadiazol-2-yl]carbamoyl]phenoxy)cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000045
cis-4-([5-[(5-benzyl-1,3,4-thiadiazol-2-yl)carbamoyl]pyridin-2-yl]oxy)cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.00012
cis-4-[4-([3-[(3,5-difluorophenyl)methyl]-1,2,4-oxadiazol-5-yl]carbamoyl)phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000011
cis-4-[4-([5-[(3,5-difluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000012
cis-4-[4-([5-[(cyclopentyloxy)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000057
cis-4-[4-[(3-benzyl-1,2,4-oxadiazol-5-yl)carbamoyl]phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000004
cis-4-[4-[(5-anilino-1,3,4-thiadiazol-2-yl)carbamoyl]phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000016
cis-4-[4-[(5-benzyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000055
cis-4-[[5-([5-[(3-chlorophenyl)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)pyridin-2-yl]oxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.25
crepidiaside C
Rattus norvegicus
-
IC50: 0.25 mM, above
0.0273
cryptotanshinone
Rattus norvegicus
-
IC50: 0.0273 mM
0.0212
dehydropipernonaline
Rattus norvegicus
-
noncompetitive inhibition, IC50: 0.0212 mM, isolated from the extracts of fruits of Piper longum and Piper nigrum
0.25
germanicol acetate
Rattus norvegicus
-
IC50: 0.25 mM, above
0.25
ixerin Y
Rattus norvegicus
-
IC50: 0.25 mM, above
0.0109 - 0.0288
kurarinone
0.0059
methyl 1-benzyl-3-[(furan-3-carbonyl)amino]-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0082
methyl 1-benzyl-3-[(furan-3-carbonyl)amino]-5-[[(thiophen-3-yl)methyl]amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0074
methyl 3-benzamido-1-[(furan-2-yl)methyl]-5-[(2-methylbutyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0091
methyl 3-[(furan-2-carbonyl)amino]-1-(3-methylbutyl)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0088
methyl 3-[(furan-3-carbonyl)amino]-1-(2-methylpropyl)-5-[(pentan-3-yl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0072
methyl 5-[(2,3-dihydro-1H-inden-2-yl)amino]-3-[(furan-3-carbonyl)amino]-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0295
methyl 5-[[(4-acetamidophenyl)methyl]amino]-1-benzyl-3-[(furan-3-carbonyl)amino]-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0192
methyl 5-[[(furan-3-yl)methyl]amino]-1-(2-methylpropyl)-3-(2-phenylacetamido)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
Homo sapiens
-
at pH 7.4 and 37°C
0.0264
methyl ursolate
Rattus norvegicus
-
IC50: 0.0264 mM
0.0035
N-(1-[[5-tert-butyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]amino]-2-methyl-1-oxopropan-2-yl)-4-fluorobenzamide
Homo sapiens
-
at pH 7.5 and 25°C
0.0085 - 0.0708
N-(4,5-dihydronaphtho[1,2-d]thiazol-2-yl)-2-(3,4-dimethoxy phenyl)acetamide
0.000048
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-(trans-4-carbamoylcyclohexyl)benzamide
Homo sapiens
-
at pH 7.4 and 37°C
0.000279
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-(trans-4-[[2-(dimethylamino)ethyl]carbamoyl]cyclohexyl)benzamide
Homo sapiens
-
at pH 7.4 and 37°C
0.000122
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-(trans-4-[[2-(morpholin-4-yl)ethyl]carbamoyl]cyclohexyl)benzamide
Homo sapiens
-
at pH 7.4 and 37°C
0.000081
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-[trans-4-[(2,3-dihydroxypropyl)carbamoyl]cyclohexyl]benzamide
Homo sapiens
-
at pH 7.4 and 37°C
0.000092
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-[trans-4-[(2-hydroxy-2-methylpropyl)carbamoyl]cyclohexyl]benzamide
Homo sapiens
-
at pH 7.4 and 37°C
0.000088
N-(5-benzyl-1,3,4-thiadiazol-2-yl)-4-[trans-4-[(2-methoxyethyl)carbamoyl]cyclohexyl]benzamide
Homo sapiens
-
at pH 7.4 and 37°C
0.000027
N-[(2S)-1-ethoxy-4-phenylbutan-2-yl]-1-[2-(tricyclo[3.3.1.1~3,7~]decan-2-yl)acetamido]cyclopentane-1-carboxamide
Homo sapiens
-
at pH 7.5 and 25°C
0.00076
N-[1,5-bis(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]-2-methyl-N~2~-[1-(trifluoromethyl)cyclopropane-1-carbonyl]alaninamide
Homo sapiens
-
at pH 7.5 and 25°C
0.000062
N-[1-(4-fluoro-2-methylphenyl)-5-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]-2-methyl-N~2~-[1-(trifluoromethyl)cyclopropane-1-carbonyl]alaninamide
Homo sapiens
-
at pH 7.5 and 25°C
0.0014
N-[1-(4-fluorophenyl)-5-[2-(4-fluorophenyl)propan-2-yl]-1H-1,2,4-triazol-3-yl]-2-methyl-N~2~-[1-(trifluoromethyl)cyclopropane-1-carbonyl]alaninamide
Homo sapiens
-
at pH 7.5 and 25°C
0.01
N-[5-tert-butyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]-2-methyl-N~2~-(1-methylcyclopropane-1-carbonyl)alaninamide
Homo sapiens
-
IC50 less than 0.01 mM, at pH 7.5 and 25°C
0.0048
N-[5-tert-butyl-1-(4-fluorophenyl)-1H-1,2,4-triazol-3-yl]-2-methyl-N~2~-[1-(trifluoromethyl)cyclopropane-1-carbonyl]alaninamide
Homo sapiens
-
at pH 7.5 and 25°C
0.0317
oleanolic acid
Rattus norvegicus
-
IC50: 0.0317 mM
0.0545
oleate
Homo sapiens
-
noncompetitive inhibition, IC50: 0.0545 mM
0.0787
phenylpyropene A
Rattus norvegicus
-
-
0.0217
phenylpyropene B
Rattus norvegicus
-
-
0.01104
phenylpyropene C
Rattus norvegicus
-
-
0.0372
pipernonaline
Rattus norvegicus
-
IC50: 0.0372 mM, isolated from the extracts of fruits of Piper longum and Piper nigrum
0.0201
piperrolein B
Rattus norvegicus
-
IC50: 0.0201 mM, isolated from the extracts of fruits of Piper longum and Piper nigrum
0.9
retrofractamide C
Rattus norvegicus
-
IC50: 0.9 mM, above, isolated from the extracts of fruits of Piper longum and Piper nigrum
0.03
roselipin 1a
Homo sapiens
-
0.04
roselipin 1B
Homo sapiens
-
0.045
roselipin 2A
Homo sapiens
-
0.05
roselipin 2B
Homo sapiens
-
0.000007
tert-butyl (2S)-2-[[1-([(2S)-2-[(2,2-dimethylpropanoyl)oxy]-4-methylpentanoyl]amino)cyclopentane-1-carbonyl]amino]-4-phenylbutanoate
Homo sapiens
-
at pH 7.5 and 25°C
0.00016
trans-4-[4-([5-[(3,5-difluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.00028
trans-4-[4-[(5-benzyl-1,3,4-thiadiazol-2-yl)carbamoyl]phenoxy]cyclohexane-1-carboxylic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.0188 - 0.0491
tussilagone
0.0992
tussilagonone
Rattus norvegicus
-
-
0.04
xanthohumol
Homo sapiens
-
0.0000014 - 0.001499
XP620
0.000019
[(1r,4r)-4-[4-(4-amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)phenyl]cyclohexyl]acetic acid
Homo sapiens
pH 7.4, temperature not specified in the publication
0.000157
[(1r,4r)-4-[4-(5-[[6-(trifluoromethyl)pyridin-3-yl]amino]pyridin-2-yl)phenyl]cyclohexyl]acetic acid
Homo sapiens
pH 7.4, 25°C
0.00008
[(1r,4r)-4-[4-(6-carbamoyl-3,5-dimethylpyrazin-2-yl)phenyl]cyclohexyl]acetic acid
Homo sapiens
pH 7.4, temperature not specified in the publication
0.000398
[4-(4-[4-[(naphthalene-2-carbonyl)amino]phenyl]thieno[3,2-d]pyrimidin-7-yl)cyclohexyl]acetic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
0.000121
[4-[4-(4-[[(3-chlorophenyl)carbamoyl]amino]phenyl)thieno[3,2-d]pyrimidin-7-yl]cyclohexyl]acetic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
1
[4-[4-(4-[[(4-chloropyridin-2-yl)carbamoyl]amino]phenyl)thieno[3,2-d]pyrimidin-7-yl]cyclohexyl]acetic acid
Homo sapiens
above, pH 7.4, 25°C
1
[4-[4-(4-[[(5-bromopyridin-3-yl)carbamoyl]amino]phenyl)thieno[3,2-d]pyrimidin-7-yl]cyclohexyl]acetic acid
Homo sapiens
above, pH 7.4, 25°C
0.000152
[4-[4-(4-[[2-phenyl-5-(trifluoromethyl)-1,3-oxazole-4-carbonyl]amino]phenyl)thieno[3,2-d]pyrimidin-7-yl]cyclohexyl]acetic acid
Homo sapiens
pH 7.4, 25°C, recombinant enzyme in microsomes of Spodoptera frugiperda cells
0.001
[4-[4-(4-[[6-(trifluoromethyl)pyridine-3-carbonyl]amino]phenyl)thieno[3,2-d]pyrimidin-7-yl]cyclohexyl]acetic acid
Homo sapiens
above, pH 7.4, 25°C
0.000019
[trans-4-(4-[[5-(2-cyclopentylethyl)-1,3,4-thiadiazol-2-yl]carbamoyl]phenyl)cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000009
[trans-4-[4-([5-[(3,5-difluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenyl]cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.00139
[trans-4-[4-([5-[(4-fluorophenyl)methyl]-1,3,4-oxadiazol-2-yl]carbamoyl)phenyl]cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.0006
[trans-4-[4-([5-[(4-fluorophenyl)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenyl]cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000038
[trans-4-[4-([5-[(cyclopentyloxy)methyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenyl]cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000144
[trans-4-[4-([5-[2-(oxolan-2-yl)ethyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenyl]cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
0.000233
[trans-4-[4-([5-[2-(oxolan-3-yl)ethyl]-1,3,4-thiadiazol-2-yl]carbamoyl)phenyl]cyclohexyl]acetic acid
Homo sapiens
-
at pH 7.4 and 37°C
additional information
amidepsine C
-
0.047
7beta-(3-ethyl-cis-crotonoyloxy)-1alpha-(2-methylbutyryloxy)-3,14-dehydro-Z-notonipetranone
Rattus norvegicus
-
-
0.1607
7beta-(3-ethyl-cis-crotonoyloxy)-1alpha-(2-methylbutyryloxy)-3,14-dehydro-Z-notonipetranone
Homo sapiens
-
-
0.211
8-angeloyloxy-3,4-epoxy-bisabola-7(14),10-dien-2-one
Rattus norvegicus
-
-
0.2944
8-angeloyloxy-3,4-epoxy-bisabola-7(14),10-dien-2-one
Homo sapiens
-
-
0.04
amidepsine A
Homo sapiens
-
0.07
amidepsine A
Homo sapiens
-
0.03
amidepsine B
Homo sapiens
-
0.06
amidepsine B
Homo sapiens
-
0.02
amidepsine D
Homo sapiens
-
0.03
amidepsine D
Homo sapiens
-
0.0098
kuraridin
Rattus norvegicus
-
-
0.0098
kuraridin
Rattus norvegicus
-
IC50: 0.0098 mM
0.0109
kurarinone
Rattus norvegicus
-
-
0.0288
kurarinone
Homo sapiens
-
-
0.0085
N-(4,5-dihydronaphtho[1,2-d]thiazol-2-yl)-2-(3,4-dimethoxy phenyl)acetamide
Homo sapiens
pH not specified in the publication, temperature not specified in the publication
0.0708
N-(4,5-dihydronaphtho[1,2-d]thiazol-2-yl)-2-(3,4-dimethoxy phenyl)acetamide
Homo sapiens
pH not specified in the publication, temperature not specified in the publication
0.0188
tussilagone
Rattus norvegicus
-
-
0.0491
tussilagone
Homo sapiens
-
-
0.0000014
XP620
Mus musculus
-
substrate: 1-hexadecanol
0.0000027
XP620
Mus musculus
-
substrate: sn-2-monooleoylglycerol
0.0000029
XP620
Rattus norvegicus
-
substrate: sn-2-monooleoylglycerol
0.0000166
XP620
Homo sapiens
-
substrate: sn-2-monooleoylglycerol
0.0000233
XP620
Homo sapiens
-
substrate: 1-hexadecanol
0.000123
XP620
Mus musculus
-
substrate: 1,2-dioleoyl-sn-glycerol
0.000176
XP620
Rattus norvegicus
-
substrate: 1,2-dioleoyl-sn-glycerol
0.001499
XP620
Homo sapiens
-
substrate: 1,2-dioleoyl-sn-glycerol
additional information
amidepsine C
Homo sapiens
IC50 above 0.2 mM
-
additional information
amidepsine C
Homo sapiens
IC50 above 0.2 mM
-
additional information
amidepsine C
Homo sapiens
-
IC50 above 0.2 mM
-
additional information
additional information
Homo sapiens
-
IC50 value for tussilagonone above 0.5 mM
-
additional information
additional information
Rattus norvegicus
-
kurarione IC50: 0.0048 mg/ml, 8-prenylleutone IC50: 0.015 mg/ml, auriculatin IC50: 0.0072 mg/ml, erysenegalensein O IC50: 0.0011 mg/ml, erysenegalensein D IC50: 0.0015 mg/ml, erysenegalensein N: 28% inhibition at 0.0125 mg/ml, derrone IC50: 0.0151 mg/ml, alpinumisoflavone: 23% inhibition at 0.0125 mg/ml, 6,8-diprenylgenistein IC50: 0.0067 mg/ml
-
additional information
roselipin 1a
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 1a
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 1a
Homo sapiens
-
IC50 above 0.2 mM
additional information
roselipin 1B
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 1B
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 1B
Homo sapiens
-
IC50 above 0.2 mM
additional information
roselipin 2A
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 2A
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 2A
Homo sapiens
-
IC50 above 0.2 mM
additional information
roselipin 2B
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 2B
Homo sapiens
IC50 above 0.2 mM
additional information
roselipin 2B
Homo sapiens
-
IC50 above 0.2 mM
additional information
XP620
Homo sapiens
-
IC50 above 0.03 mM with 1,2-dioleoyl-sn-glycerol or sn-2-monooleoylglycerol as substrate